Meldonium: umarnin don amfani, alamomi don amfani da softronate

Ana samun Mildronate a cikin nau'ikan sashi na gaba:

  • Capsules: farar fata, gelatin mai wuya, girman No. 1 (250 MG) ko No. 00 (500 MG), abinda ke cikin capsules shine farin farin hygroscopic crystalline farin foda tare da wari mara kyau (a cikin blisters na 10 inji., 2, 4, 6 ko blisters a cikin wani kwali mai kwali),
  • Magani don allura: mara launi, m (a cikin ampoules na 5 ml, 5 ampoules a cikin blisters, fakitoci 2 a cikin kwali na kwali).

Abun da ke ciki na capsule 1 ya hada da:

  • Abunda yake aiki: meldonium dihydrate - 250 ko 500 MG,
  • Abubuwan taimako: sitaci dankalin turawa - 13.6 / 27.2 mg, colloidal silicon dioxide - 5.4 / 10.8 mg, alli stearate - 2.7 / 5.4 mg.

Abun da ke ciki na kwanson kwalliya: E171 (titanium dioxide) - 2%, gelatin - har zuwa 100%.

Tsarin 1 ml na bayani ya haɗa:

  • Abubuwan da ke aiki: meldonium - 100 MG (a cikin nau'in propimate na trimethylhydrazinium),
  • Bangaren taimako: ruwa don yin allura.

Alamu don amfani

  • Rage yawan aiki, ƙwayar jiki (gami da athletesan wasa),
  • Cutar Abastinence a cikin na kullum na shan giya (lokaci guda tare da takamaiman magani don shan giya),
  • Cututtukan zuciya da na jijiyoyin jini (myocardial infarction, minacardial infarction, angina pectoris), gajiyawar zuciya (a zaman wani yanki na hadaddun jiyya),
  • Cutar cuta mai saurin kamuwa da cuta da rashin aiki ta hanji, gami da shanyewar jiki da kuma karancin hancin ciki (a zaman wani bangare na hadaddun jiyya).

Additionallyarin ƙari don Mildronate a cikin nau'i na mafita don allura:

  • Thrombosis daga cikin jijiya na tsakiya da kuma rassan sa,
  • Hemophthalmus, retinal basur na daban-daban etiologies,
  • Retinopathies na daban-daban etiologies (hauhawar jini, masu ciwon sukari).

Contraindications

  • Pressureara yawan matsa lamba cikin mahaifa (gami da ciwan ciki, daɗaɗɗar gurɓataccen ruwan ciki),
  • Rashin hankali ga miyagun ƙwayoyi.

Bayar da magunguna ga yara 'yan ƙasa da shekaru 18, da kuma masu shayarwa da mata masu juna biyu, ba a ba da shawarar saboda rashin bayanan asibiti wanda ke tabbatar da amincin da tasirin Mildronate a cikin waɗannan rukunin marasa lafiya.

Ya kamata a yi amfani da Mildronate tare da taka tsantsan a cikin marasa lafiya da cututtuka na kodan da / ko hanta (musamman na dogon lokaci).

Sashi da gudanarwa

Sakamakon yiwuwar haɓaka sakamako mai ban sha'awa, ana bada shawarar yin amfani da Mildronate a farkon rabin rana, lokacin ɗauka sau da yawa a rana - ba tare da ƙarfe 17.00.

A ciki, Mildronate a cikin kwalliyar kwalliya galibi ana wajabta shi kamar haka:

  • Cututtukan zuciya da na jijiyoyin zuciya (myocardial infarction, angina pectoris), gajiyawar zuciya: kashi na yau da kullun - 500-1000 MG, mita na gudanarwa - sau 1-2 a rana. Tsawon lokacin karatun warkewa shine watanni 1-1.5 (a lokaci guda tare da wasu kwayoyi),
  • Dyshormonal cardiomyopathy: kashi na yau da kullun - 500 MG. Tsawon lokacin aikin warkewa shine kwanaki 12 (lokaci guda tare da wasu kwayoyi),
  • Hatsarori na Subacute cerebrovascular (karancin ƙwayoyin cerebrovascular insufficiency da bugun jini): kashi na yau da kullun - 500-1000 MG, mita na gudanarwa - sau 1-2 a rana. Tsawon lokacin karatun warkewa shine watanni 1-1.5 (ana ɗaukar maganin a baki a lokaci ɗaya kamar sauran kwayoyi bayan ƙarshen aikin allura tare da Mildronate),
  • Hatsari na ƙwayar cuta na yau da kullun: kashi na yau da kullun - 500 MG. Tsawon lokacin aikin warkewa shine watanni 1-1.5 (lokaci guda tare da wasu kwayoyi). Yana yiwuwa a gudanar da maimaita karatun (galibi sau 2-3 a shekara) bayan shawarwarin likita,
  • Rage yawan aiki, ƙwaƙwalwar tunani da ta jiki (ciki har da tsakanin masu motsa jiki): kashi ɗaya na yau da kullun - 1000 mg, mita na gudanarwa - sau 2 a rana. Tsawon lokacin aikin warkewa shine kwanaki 10-14. Bayan makonni 2-3, hanya ta biyu tana yiwuwa,
  • Cutar da mutum cikin cututtukan shan barasa: kashi biyu a kowace rana na milimita 2000, yawan gudanarwa - sau 4 a rana. Tsawon lokacin aikin warkewa shine kwanaki 7-10 (a lokaci guda tare da takamaiman maganin shan barasa).

'Yan wasan motsa jiki kafin horo suna da shawarar shan Mildronate a kashi daya na 500-1000 MG sau 2 a rana. Tsawon lokacin karatun a cikin lokacin shiri shine makonni 2-3, yayin lokacin gasa - ranakun 10-14.

Mildronate a cikin hanyar samar da mafita don allura ana gudanar dashi a cikin jijiya da parabulbarno.

A matsayinka na mai mulkin, an wajabta magani mai guba

  • Cutar cututtukan zuciya: kashi na yau da kullun - 500-1000 MG (5-10 ml na maganin allura, taro - 500 MG / 5 ml), yawan amfani 1-2 sau a rana. Tsawon lokacin karatun shine watanni 1-1.5 (a lokaci guda tare da wasu kwayoyi),
  • Haɗarin Cerebrovascular (lokaci mai ƙarfi): kashi ɗaya na yau da kullun - 500 MG, yawan amfani - lokaci 1 a rana. Ana gudanar da maganin don kwanaki 10, bayan haka sun canza zuwa shan Mildronate na baki (500-1000 MG kowace rana). Jimlar lokacin aikin magani shine watanni 1-1.5,
  • Damuwa ta jiki da ta hankali: kashi na yau da kullun - 500 mg, yawan amfani - lokaci 1 a rana. Adadin aikin jiyya shine kwana 10-14. Bayan makonni 2-3, hanya ta biyu tana yiwuwa,
  • Shan giya na yau da kullun: maganin yau da kullun - 1000 mg, yawan amfani - sau 2 a rana. Adadin aikin jiyya shine kwana 10-14.

Game da cututtukan jijiyoyin jiki da cututtukan dystrophic na retina, ya kamata a gudanar da Mildronate parabulbarly a cikin kashi na 0.5 ml na maganin allura tare da taro na 500 MG / 5 ml na kwanaki 10.

Side effects

A cikin lokuta mafi wuya, tare da yin amfani da Mildronate a duk siffofin sashi, irin wannan sakamako na iya haifar da haɓaka kamar: halayen rashin lafiyan (itching, redness da fata, urticaria, fatar fata, angioedema), dyspepsia, tachycardia, ƙara ko rage karfin jini, haɓaka haushi.

A cikin lokuta mafi wuya, ci gaban eosinophilia da rauni gaba ɗaya yana yiwuwa.

Hulɗa da ƙwayoyi

Tare da amfani da lokaci guda na Mildronate tare da wasu kwayoyi, sakamakon da ba a ke so ba na iya faruwa:

  • Magungunan kwantar da hankali na hanji, wasu magungunan antihypertensive, cardiac glycosides: haɓaka aikin su,
  • Nitroglycerin, nifedipine, alpha-adrenergic blockers, magungunan antihypertensive da magungunan jijiyoyi: haɓakar jijiyoyin jini, tachycardia matsakaici (yakamata a yi taka tsantsan lokacin amfani da irin waɗannan haɗuwa).

Ana iya tsara Mildronate lokaci guda tare da tsawan tsawan nau'ikan nitrates, sauran magungunan antianginal, jami'in antiplatelet da maganin anticoagulants, antiarrhythmic, bronchodilator da magungunan diuretic.

Halayen magunguna

An tsara waɗannan magungunan don karuwar motsa jiki, tsananin wasanni da raunin ƙwaƙwalwar ajiya da taro.

Tare da cututtukan zuciya da ischemia, yana mayar da isar da oxygen zuwa sel. Increara aikin tunani da ta jiki, yana kawar da tasirin damuwa na kwakwalwa, yana da tasirin zuciya.

Ana amfani da miyagun ƙwayoyi don gazawar zuciya da kuma magance cututtukan cututtukan fata. Siffar saki - capsules da mafita don allura.

Hakanan maganin yana kara karfin garkuwar jiki da juriya ga damuwa.

Magungunan yana gajarta lokacin murmurewa bayan bugun zuciya, yana taimakawa rage yankin necrosis.

Magungunan yana taimakawa rage yawan cututtukan angina. Ana amfani dashi don ƙara ƙarfin hali a cikin 'yan wasa. Zata iya bada tabbatacciyar amsawa game da gwajin doping. Magungunan yana taimakawa haɓaka kwararar jini zuwa wurin ischemia, wanda ke hanzarta dawo da yankin da cutar ta shafa.

Mildronate yana taimakawa rage yawan faruwar cutar angina.

An wajabta magungunan don cututtukan cututtukan cuta wanda ke faruwa a cikin asusun. Magungunan yana da tasirin tonic, saboda haka ana bada shawara don amfani dashi da safe. An wajabta maganin don maganin ciwon sukari azaman adjuvant.

Kwatanta Meldonium da Mildronate

Magungunan suna da kamala iri ɗaya kuma abu mai aiki - meldonium dihydrate. Alamu don amfanin magunguna biyu:

  • cututtuka na tsarin zuciya da jijiyoyin jini,
  • rikicewar Sistem a cikin kwakwalwa,
  • karban ciwo a cikin marasa lafiya da na kullum shan giya,
  • nauyi mai nauyi da damuwa na jiki,
  • ilimin cututtukan fata,
  • lokacin murmurewa bayan tiyata.

Contraindications ma iri ɗaya ne ga duka magunguna:

  • hawan jini
  • lokacin shayarwa da ciki,
  • yara 'yan ƙasa da shekara 18,
  • pressureara yawan matsa lamba na ciki.

Side effects na kwayoyi iri daya ne:

  • abubuwan dyspeptik
  • karuwa a cikin jini,
  • bugun zuciya
  • alerji

Wanda ya kirkiro magungunan duka shine Vidal. Kada a haɗu da magunguna tare da alpha-blockers da nitroglycerin. In ba haka ba, bayyanar tachycardia mai yiwuwa ne. Ana amfani da magunguna biyu tare da taka tsantsan a cikin cututtukan koda da na hanta.

Menene kamancecennin magungunan:

  • iri ɗaya aiki
  • guda pharmacological sakamako
  • nau'ikan jerin abubuwan contraindications da sakamako masu illa,
  • daya kamfanin.

Menene Meldonium don? Umarnin, farashi da bita

A cikin wannan labarin na likita, zaku iya samun masaniya da miyagun ƙwayoyi Meldonium. Umarnin don amfani zai yi bayani a cikin waɗanne lokuta zaka iya ɗaukar kwayoyin magani da allura, abin da magunguna ke taimaka wa, menene alamun akwai amfani, maganin hana haifuwa. Bayanin yana gabatar da kamannin magungunan da abubuwan da ya ƙunsa.

Maganin anti-arrhythmic na aji na IB, inganta metabolism - tafiyar matakai na rayuwa a jikin mutum shine Meldonium. Umarnin don amfani yana ba da shawarar ɗaukar capsules ko allunan 250 MG da 500 MG, injections a cikin ampoules don allura don lura da haɗarin cerebrovascular, dawo da ƙarfi a cikin 'yan wasa, cututtukan zuciya na ischemic.

Mahimmanci! An san Meldonium a matsayin mai dope. An hana amfani dashi a cikin wasanni masu sana'a!

Kayan magunguna

Hanyoyin haɓaka ƙwayar cuta, anama gamma-butyrobetaine. Yana hana gamma-butyrobetaine hydroxynase, yana hana haɗin carnitine da jigilar daskararren sarkar acid ta hanyar membranes, kuma yana hana tara nau'ikan kitse na unoxidized mai mai a cikin sel - abubuwan da ke faruwa na acylcarnitine da acylcoenzyme A.

A karkashin yanayin ischemia, yana dawo da daidaituwa na tafiyar matakai na isar da oxygen da yawan amfani da shi a cikin sel, yana hana cin zarafin jigilar jigilar ATP, kuma a lokaci guda yana kunna glycolysis, wanda ke gudana ba tare da ƙarin amfani da oxygen ba.

Sakamakon raguwa a cikin taro na carnitine, gamma-butyrobetaine tare da kaddarorin vasodilating yana haɓaka mai ƙarfi. Hanyar aiki yana ƙayyade bambancin tasirin magunguna: haɓaka haɓaka, rage alamun damuwa da damuwa na jiki, kunna nama da rigakafin ƙwaƙwalwar mutum, tasirin cutar zuciya.

Tasiri

Game da mummunar cutar ischemic a cikin myocardium, yana rage jinkirin samuwar yankin necrotic kuma yana gajarta lokacin murmurewa. Tare da rashin karfin zuciya, yana kara yawan kwanciyar hankali na mutum, yana kara karfin motsa jiki, da kuma rage yawan kamuwa da cutar angina.

A cikin mummunar cuta da rashin lafiyar ischemic na wurare dabam dabam na haɓakar cerebral yana inganta wurare dabam dabam na jini a cikin ischemia, yana ba da gudummawa ga sake rarraba jini a madadin yankin ischemic. Inganci ga cututtukan jijiyoyin bugun gini da na dystrophic na fundus.

Yana da sakamako na tonic akan tsarin juyayi na tsakiya, yana kawar da rikice-rikice na aiki na tsarin juyayi a cikin marasa lafiya tare da shan barasa tare da ciwo na cirewa.

Menene Meldonium don?

Manuniya don amfani sun haɗa da hadadden far:

  • kangin aiki,
  • karban ciwo a mahaukaci,
  • Ciwon zuciya,
  • rage aiki
  • hatsarori na ciki,
  • dishormonal cardiomyopathy,
  • Gyaran bayan aikin asibiti

Abin da Parabulbar gwamnatin taimaka daga:

  • retinal thrombosis,
  • retinopathies (masu ciwon sukari da hauhawar jini),
  • bashin ciki
  • cuta na cikin jijiyoyin hannu a cikin retina.

Umarnin don amfani

An bada shawarar Meldonium da safe, saboda yana iya haifar da sakamako mai ban sha'awa. An saita kashi ɗaya akayi daban-daban dangane da alamun da kuma hanyar gudanarwa.

Lokacin ɗauka ta baki, kashi ɗaya shine 0.25-1 g, yawan sarrafawa da tsawon lokacin jiyya yana dogara ne da alamun.

0.5 ml na allurar bayani tare da maida hankali ne akan 500 MG / 5 ml ana gudanar da shi a cikin layi ɗaya na kwana 10.

Tare da gudanarwa na ciki, kashi shine 0.5-1 g 1 lokaci kowace rana, tsawon lokacin jiyya yana dogara da alamun.

An wajabta wa 'yan wasan motsa jiki don warkewar motsa jiki bisa ga tsarin musamman a hade tare da wasu hanyoyi. A bisa hukuma an yarda da shi azaman goro.

Yadda za a ɗauka tare da cututtuka?

  1. Game da yaduwar illa, ana bada shawarar Meldonium a lokacin ɓarkewar 0.5 g sau ɗaya a rana don kwanaki 10, to a cikin nau'in encapsulated - 0.5 g kowace rana don kwanakin 14-21.
  2. A cikin yanayin da ke fama da haɗarin kamuwa da cuta na ƙwaƙwalwar ƙwayar cuta, an tsara hanya ta jiyya ta tsawon kwanaki 14-21. Ana gudanar da allurar rigakafin intramuscularly a 0.5 g sau ɗaya a rana ko ana gudanar da shi a baki a 0.25 g (mita na sarrafawa ya dogara da tsananin yanayin yanayin mai haƙuri).
  3. Rashin ciwo yana buƙatar hanya na magani tare da Meldonium na kwanaki 7-10. Sannan za a nuna mai haƙuri sau hudu na miyagun ƙwayoyi a lokacin rana, 0.5 g a ciki ko na lokaci-lokaci biyu.
  4. Tare da barga angina pectoris, kwanakin 3-4 na farko ana wajabta su sau 0.25 g sau 3. Sannan ana shan su a baki sau biyu a sati a sati sau 0.25 g sau 3. Tsawan lokacin jiyya daga 4 zuwa 6 ne.
  5. Tare da cardialgia, tare da dishormonal myocardial dystrophy, ana gudanar da maganin a cikin hanyar jet sau ɗaya a rana, 0.5-1 g ko IM har zuwa sau 2 a rana, 0.5 g. 0.25 MG da safe da maraice, ana ci gaba da jinya don wani kwanaki 12.
  6. Tare da rashin daidaitaccen nau'in angina pectoris da infarction na myocardial, ana amfani da Meldonium a cikin jijiya ta hanyar jet na 0.5 g ko 1 g sau ɗaya a rana. Bayan haka, an wajabta shi a baki: 3-4 days - 0.25 g sau 2, sannan 2 days a mako 0.25 g sau 3 a rana.
  7. Idan akwai cututtukan jijiyoyin jiki daga cikin asushin, dystrophy na retinal, Meldonium an wajabta shi a kan abin da ya faru na 10,05 g a cikin kwanaki 10.
  8. A cikin rauni na zuciya, ana gudanar da maganin a cikin jijiya a cikin kullun a kashi na 0.5-1 g ko an maye gurbinsu da allurar intramuscular na 0.5 g har sau 2 a rana. Bayan kwanaki 10-14 na jiyya, an tura mai haƙuri zuwa cajin gg 0,5, wanda yakan dauki lokaci 1 da safe. Hanyar magani daga makonni hudu zuwa shida ne.

Karanta wannan labarin: Ademethionine

Yara yayin daukar ciki da lactation

Ba a tsara Meldonium ga mata masu juna biyu ba, tunda ba zai yiwu a tabbatar da lafiyar mahaifiyar da jaririn ba. Idan kuna buƙatar rubuta magani don mace mai shayarwa, to, a lokacin jiyya, an dakatar da shayarwa: ba a san ko kayan zai shiga cikin madara ba.

A cikin yara da matasa masu shekaru 18, ba a kafa ingantaccen tasiri da amincin lafiyar meldonium ba. Meldonium a cikin nau'i na capsules an contraindicated don amfani a cikin yara da matasa a ƙarƙashin shekara 18, a cikin nau'i na syrup a cikin yara a ƙarƙashin shekaru 12.

Umarni na musamman

Yi amfani tare da taka tsantsan a cikin cututtukan hanta da / ko kodan, musamman na dogon lokaci.

Shekaru da yawa na gogewa a cikin lura da matsanancin ƙwayar cuta na zuciya da rashin angina a cikin sassan aikin zuciya yana nuna cewa meldonium ba shine farkon layin farko na cututtukan jijiyoyin zuciya ba.

Haɗa kai

Tare da yin amfani da lokaci ɗaya tare da Nitroglycerin, alpha-blockers, Nifedipine, vasodilators na gefe, akwai yiwuwar tachycardia da hypotension arterial. Yana inganta aikin antihypertensive, magungunan antianginal, glycosides na zuciya.

Wataƙila haɗuwa tare da magungunan antianginal, maganin anticoagulants, magungunan antiarrhythmic da diuretics.

Mahimmanci! Karka yi amfani dasu lokaci guda tare da wasu magunguna waɗanda ke ɗauke da meldonium.

Analogs na miyagun ƙwayoyi Meldonium

Tsarin yana tantance analogues:

  1. Vasomag.
  2. Meldonium bushewa.
  3. Idrinol
  4. Meldonium Organics (Binergia, Eskom).
  5. Angiocardyl.
  6. 3- (2,2,2-Trimethylhydrazinium) daskararru.
  7. Cardionate
  8. Midolat.
  9. Medatern.
  10. Tafiya.
  11. Mildronate

Don lura da nauyin jiki da na tunani, dawo da jiki, ana analo analogues ta aiki:

  1. Lamivit.
  2. Eleutherococcus cirewa.
  3. Harshen Cigapan.
  4. Yantavit.
  5. Falkamine.
  6. Ascovite.
  7. Galavit.
  8. Centrum.
  9. Cardionate
  10. Bashin
  11. Hepargin.
  12. Triovit.
  13. Idrinol
  14. Eltacin.
  15. Corilip.
  16. Ribonosin
  17. Vazoton (L-arginine).
  18. Vasomag.
  19. Selmevit.
  20. Pikovit forte.
  21. Berocca da.
  22. Pantogam.
  23. Heptolexin.
  24. Mildronate
  25. Abincin abinci.
  26. Litattafan mahaifa Ubiquinone.
  27. Valeocor Q10.
  28. Pikovit.
  29. Kudewita.
  30. Carnitine.
  31. Dibikor.
  32. Trekrezan.
  33. Abinci.
  34. Elkar.
  35. Riboxin
  36. Vitamax
  37. Harshen Pantocalcin.
  38. Antioxidants tare da aidin.
  39. Cytoflavin.
  40. Harshen Cropanol.
  41. Neoton.
  42. Nagipol.
  43. Bashin
  44. Jeriton.
  45. Oligovit.
  46. Duovit.
  47. Encephabol.
  48. Kudesan.
  49. Metaprot.
  50. Withara tare da baƙin ƙarfe.
  51. Asvitol.
  52. Inosine.
  53. Vitrum ƙari.
  54. Leriton kadari.
  55. Saukad da Beresh ƙari.
  56. Coenzyme compositum.

Sharuɗɗan hutu da farashi

Matsakaicin farashin Meldonium (injections na 5 ml No. 10) a cikin Moscow shine rubles 145. A cikin Ukraine, zaku iya siyan magani don hryvnia na 195. a cikin Kazakhstan, kantin magunguna suna ba da alamar analog of Mildronate. A cikin Minsk, suna sayar da maganin don bel bel. rubles. Don samun magani, kuna buƙatar takardar sayan magani.

Ta hanyar bin hanyoyin haɗin, zaka iya gano wannene analogues don amfani da cututtukan cututtukan: cirewar bayyanar cututtuka, shan giya, hemophthalmus, dishormonal cardiomyopathy, bugun jini, myocardial infarction, hemorrhage, angina pectoris, thrombosis, tashin hankali na jiki, gajiyawar zuciya, gazawar zuciya

Mildronate - yadda ake ɗaukar 'yan wasa

An gano Meldonium a cikin karni na 70 na karni na 20 a Cibiyar Nazarin Kwayoyin ta Latvian kuma an fara amfani dashi azaman mai haɓaka shuka da dabbobi, kuma daga baya aka fara amfani dashi a cikin yanayin kiwon lafiya. Bayan lokaci, likitoci sun fara tsara shi don cututtuka daban-daban a matsayin wakili na rayuwa kuma suna ba da shawara ga 'yan wasa don murmurewa mafi kyau.

Me yasa ake buƙatar meldonium a wasanni

Mene ne ƙaramin abu, kuma yan koyo zasu iya ɗaukarsa? Maganin shine kwatancin wucin gadi na gamma-butyrobetaine - enzyme da aka samo a cikin kowane sel na jikin mutum.

Hanyar aiwatar da maganin. Meldonium yana toshe samar da carnitine a cikin jiki yana rage jinkirin amfani da mai mai a matsayin tushen kuzari. Yawancin lokaci shine cincin da aka cinye lokacin da mutane ke cinye makamashi wanda ke jagorantar rayuwa mai aiki.

Kuma ana canza mayukan kitse zuwa makamashi a cikin kwayoyin halittar tsoka, wanda ke sanya zuciya yin aiki a hanzari. Ayyukan matsakaita shine sake ginawa da canzawa zuwa samar da makamashi daga glucose da oxygen. Wannan yana rage nauyi a zuciya da sauran gabobin jiki.

A cikin aikinsa, miyagun ƙwayoyi shine kishiyar mai ƙari kamar L-carnitine.

Babban maƙasudin Mildronate shine haɓaka metabolism da jikewar kuzari a matakin salula.

M kaddarorin amfani na meldonium a wasanni

  • Yana saurin murmurewa bayan ƙoƙarin jiki. Kayan yana dacewa da kowane wasa, a cikin dakin motsa jiki yana iya zama duka cardio da horo mai ƙarfi. Abubuwan da aka keɓe sun kasance mafi sauri daga sel, kuma hanyoyin dawowa suna ci gaba cikin yanayin hanzari. Sakamakon haka, mai motsa jiki na iya horar da mafi yawan lokuta kuma ya ƙaru.
  • Yana kwantar da halayen jiki ga juyayi da yawan aiki na jiki. Wannan tasirin softronate zai zama da amfani musamman yayin gasa ko bushewa, lokacin da dukkanin albarkatun jiki ke lalacewa da sauri.
  • Ayyukan gaba ɗaya yana ƙaruwa kuma yawan farashi yana ƙaruwa. Mai wasan motsa jiki ya zama mafi tsufa, yana ƙaruwa, yana ƙaruwa da motsi da kuma yawan damuwa.
  • Yana haɓaka jigilar glucose zuwa sel kuma yana kiyaye zuciya daga arrhythmias, angina pectoris. Wannan shine rigakafin kamuwa da cutar cututtukan zuciya kamar bugun zuciya ko bugun jini.
  • Da amfani ga asthenia. Shan maganin yana ba ku damar kawar da ciwo na gajiya, rashin ƙarfi da rauni. Duk wannan, hakika, yana da tasirin gaske game da sakamakon wasanni.

Ana iya amfani da Meldonium don kowane nau'in kaya a cikin dakin motsa jiki. Koyaya, bai kamata kuyi tsammani ba bayan ɗaukar haɓakar alamun ƙarfin da sauri saurin ƙwayar tsoka. Wannan ƙwayar ba ta shafi ci gaban ƙwayar tsoka ta kowace hanya, kuma idan an sami ƙarin ƙaruwa a cikin ƙarfi, to, yana da ƙima sosai.

A mataki na samun riba mai yawa kuma cikin ƙarfin ƙarfi, ya cancanci amfani da meldonium kawai don mafi kyawun dawo da haɓaka ƙarfin jiki.

Mildronate zai zama mafi inganci yayin tsawan motsa jiki na motsa jiki. An wajabta wa masu tsere, 'yan wasan ƙwallon ƙafa, daskararru don juriya da haɓaka sautin zuciya. Yana kare yan wasa daga wuce gona da iri.

Kowa ya san abin da ya faru lokacin da ɗan tsere ya sami rauni a lokacin gasar, saboda jiki ba zai iya tsayar da ɗaukar nauyinsa ba.

Amfani da meldonium yana guje wa yanayi mai haɗari ga lafiya.

Idan kun kasance a kan tsayayyen abinci yayin horo mai himma, to shan Mildronate shima zai zama mai tasiri. Sakamakon ingantaccen metabolism a cikin sel, metabolism yana ƙaruwa kuma ana rasa tsari mai ƙarfi.

Koyaya, yana da mahimmanci a lura cewa ba lallai ba ne a haɗa meldonium da mai-mai mai yawa, har ma da abin da ake amfani da su na carbohydrate.

Babban tushen samar da makamashi yayin shan Mildronate shine glucose, don haka bai kamata ku rage yawan adadin carbohydrates mai sauƙi da rikitarwa ba, har ma lokacin bushewa.

Me yasa ana daukar meldonium doping

A watan Janairun 2016, Mildronate an saka shi a cikin jerin magungunan da aka haramta kuma yanzu an dauke shi bisa hukuma a matsayin doping. A waccan lokacin, wani abin kunya ya ɓarke ​​tare da 'yan wasan whoan Rasha waɗanda suka daɗe suna amfani da matsakaita.

Irin wannan farin ciki ya taka rawa a hannun masu kera meldonium, kamar yadda farashin kayayyaki ya karu sosai. A yau, tambaya game da abin da ake buƙata don ƙara motsa rai ba kawai ƙwararrun masana daga fannoni daban-daban na wasanni ba, har ma baƙi na yau da kullun zuwa wurin motsa jiki.

Har yanzu, yawancin likitoci ba su fahimci dalilin da yasa meldonium yake magana akan doping ba. Bayan duk wannan, an ƙirƙira shi musamman don tallafawa kiwon lafiya da rigakafi, babu magana game da kowane ƙaruwa na haɓaka ta iyawa ta zahiri.

Babban fasalin haramcin na Mildronate shine babban tasirinsa akan aikin dan adam, karuwa a gaba daya da kuma sakamako mai karfafa gwiwa.

Saboda waɗannan tasirin, ɗan wasa mai shan Mildronate zai sami fa'ida a gasar.

Idan kunyi wa kanku aiki, to kada kuji tsoron amfani da maganin. Amincewa da al'ada, yana da aminci ga jiki. Amma ga 'yan wasa da ke yin gasa da bayar da gudummawar jini don gwaji, yana da kyau a bar meldonium ko a yi amfani da shi tun kafin a yi.

Amfani da magani a magani

Bambancin nau'ikan maganin yana sa shi tasiri cikin cututtuka daban-daban. An wajabta Mildronate don matsaloli masu zuwa:

  • Cututtukan fata na yau da kullun, asma da sauran cututtukan cututtukan da ke tattare da numfashi,
  • Daidaitawar maganin cututtukan zuciya - angina pectoris, infarction na zuciya, rashin karfin zuciya,
  • Hadarin,
  • Tsawo wajan tunani da gajiya,
  • A matsayin magani ga m hangout da na kullum shan giya,
  • Cututtukan ido da ke hade da cuta na nakasar jini,
  • A wasu nau'ikan ciwon sukari,
  • Lokacin aikin bayan-lokaci zuwa saurin warkewa.

Duk da yawan kyawawan kaddarorin, meldonium, kamar kowane magani, yana da wasu iyakoki. Ba'a ba da shawarar ɗaukar shi ga yara 'yan ƙasa da shekaru 18 ba, yayin daukar ciki, tare da raunin craniocerebral, cututtukan fata mai lalacewa, koda, hanta, da matsalolin tsarin juyayi. Bayani mai zuwa, hanyoyin da za a iya biyo baya masu yiwuwa ne:

  • Rage saukar karfin jini
  • Rateara yawan zuciya,
  • Rashin tsayi.

Don hana sakamako masu illa, ana bada shawara don amfani da Mildronate da safe kuma kada ku ƙetare sashi. A cikin lokuta mafi sauƙi, halayen rashin lafiyan suna yiwuwa, kazalika da ƙwannafi, tashin zuciya bayan ɗauka.

Yadda ake ɗaukar meldonium don 'yan wasa

An gabatar da miyagun ƙwayoyi a cikin nau'i na capsules, Allunan da syrup, waɗanda aka yi nufin gudanar da maganin baka. Akwai kuma wani nau'in mafita wanda za'a iya gudanar dashi ta intravenously ko intramuscularly.

Yaya za a ɗauki Mildronate don 'yan wasa don samun babban aiki? Tabbas, injections na subcutaneous suna da sauri kuma sun fi tasiri.

Koyaya, a wannan yanayin, yana da mahimmanci a tsayar da lura sosai kuma yana da kwarewar allura, in ba haka ba yana iya zama cutarwa ga lafiyar. Athletesan wasan tsere na amateur sun gwammace da zaɓin kwamfutar hannu da nau'in kawa.

Lokacin da aka sha shi a baki, Mildronate ya bugu da safe rabin sa'a kafin cin abinci, ko mintuna 30 bayan cin abinci. Magungunan ba zai iya murkushewa ko tauna ba, an haɗiye shi baki ɗaya kuma an wanke shi da ruwa mai yawa.

Don haɓaka wasan motsa jiki, ana bada shawara don ɗaukar meldonium a 500 MG a rana, wato 250 mg sau 2 a rana ko 1 sau ɗaya kowace rana 500 MG. A ranar horo, ya kamata ku ɗauki abu rabin sa'a kafin aji.

Ana yin lissafin daidai gwargwadon nauyi - 15-20 a kowace kilogiram na nauyin jiki. Wa'adin ƙarshe na ƙarshe ya kamata ya kasance ba tare da ƙarshen 1700 ba ko kuma daga baya 5 hours kafin lokacin bacci don guje wa yawan damuwa.

Masu sana'a na iya haɓaka sashi sau 2 kuma suna ɗaukar kayan sau 2 a rana.

A cikin daidaitaccen kunshin, meldonium ya ƙunshi capsules 40 na 250 MG. Hakanan akwai samfuran capsule 60 na 500 MG kowane. Kudin a cikin kantin magani ya bambanta daga 230 zuwa 400 rubles.

Hakanan zaka iya samun maganin 10% na Mildronate don allura - ampoules 10 na 5 ml. Poaya daga cikin ampoule ya ƙunshi 500 MG na meldonium. Yana da mahimmanci a bi umarni kuma kada a rikita maganin matsalar cikin ciki.

Bayan buɗe ampoule, yakamata a allurar da shi nan da nan, tunda magani ba ya ƙyale saduwa da iska sama da minti 5. Kudin kunshin 1 tare da injections daga 68 zuwa 150 rubles. Tsawan lokacin ɗaukar Mildronate shine makonni 3-5.

Sannan yakamata ayi hutu na kusan wata guda don gujewa sabawa jiki. Bayan haka ana iya maimaita karatun.

"Mildronate - menene taimaka da kuma yadda ake amfani?"

Ba za a iya faɗi ba tare da karin gishiri ba cewa babu magani guda ɗaya a cikin duk tarihin zamani da aka inganta "ingantacce", haka nan, kamfanin masana'antar bai sanya ɗanɗana kuɗaɗe a kamfen tallan duniya ba. Muna magana ne game da jerin maganganun doping a cikin "babban wasanni" wanda meldonium (INN), kamar yadda ake kira shi a ƙasashen waje, ko Mildronat, kamar yadda ake kira shi a Rasha (sunan kasuwanci), ya kasance abin zargi.

Dukkanin sun fara ne a Janairu 1 na ƙarshe, 2016. A lokacin ne WADA (Hukumar Kula da Duniya ta Duniya) ta gabatar da meldonium, aka Mildronat, a cikin jerin kudaden da aka hana.

Dalilin shine gaskiyar cewa tasirin cytoprotective da sakamako na rayuwa na iya (da tsammanin) canza myocardium sosai har zuciya zata zama mai juriya da ƙarfi sosai, wanda zai sa ya yiwu a cimma nasara, sabili da haka ana samun kuɗi masu yawa.

Tarihin wannan magani yana daɗaɗɗa.

An fara kirkiro shi ne a cikin Latvian SSR ta Ivars Kalvins, kuma da farko suna son amfani da shi don zubar da kayan mai guba na man roka (dimethylhydrazine).

Amma lokacin da ake nazarin yawan guba da wannan ƙwayar a cikin dabbobi, an gano irin waɗannan sakamakon cewa tun 1976, an yi rajistar wani magani da ake kira Mildronate a cikin USSR, sannan kuma a Amurka (tun 1984).

Ba a san dalilin da yasa ba, amma a Amurka magungunan "maras kyau" ne: a cikin shekarun 80s na karni na karshe an haramta shi. A cikin ƙasarmu, amfani da allunan Mildronate ya fara a cikin magungunan soja, sannan, bayan rushewar USSR, ya zama magungunan da aka fi amfani da shi a cikin aikin likita na yau da kullun.

Abubuwa da tsarin aiwatarwa

Mildronate hoto na capsules da bayani don injections

Magungunan yana aiki akan ƙwayar zuciya ta hanyar metabolism na kitse mai. Sakamakon haka, tattarawar samfuran sinadarin oxidized a cikin sel na myocardial - myocardiocytes - yana raguwa, kuma damar yiwuwar iskar shaka mara nauyi ta ragu. Yawancin lokaci, duk waɗannan abubuwa suna tsoma baki tare da jigilar kayayyaki na ATP - kwayar halitta ta duniya - "baturin", wanda ke ba da dukkanin ƙwayoyin da makamashi.

Sakamakon haka, myocardiocytes sun sami damar yin amfani da glucose mafi kyau, kuma ana haɓaka samar da makamashi na myocardial. Kuma wannan kai tsaye yana haifar da gaskiyar cewa zuciya tana yin nasara da kyau tare da ƙara nauyin. Bugu da ƙari, ATP ba kawai aiki bane a cikin myocardium.

Groupsungiyoyi da yawa na masana kimiyya sun gano cewa miyagun ƙwayoyi suna maganin lafiya idan jiki dole yayi aiki a cikin yanayin hypoxia na salula. Mildronate yana haɓaka saurin dawowa bayan aiki mai nauyi, gami da dawo da hankalin-tunanin rai.

Magungunan suna ba da damar 'yan wasa su ba da kansu kawai gwargwadon damar su kuma "ba da mafi kyawun" a cikin horo. Koyaya, ba kwayoyin bane, ba shi da tasiri na anabolic, kuma baya haifar da ginin tsoka. Yana hana lalacewar zuciya, da inganta jijiyoyin jini, kuma yana hana cutar kwakwalwa.

Alamu da siffofin sakin

Me ke taimaka wa Mildronate? A zahiri, takaddara mai aiki (wanda, a tsakanin sauran abubuwa, WADA kuma an karkatar da shi) koyarwa ce don amfani. Shahararrun fitattun nau'ikan saki sune 250 da kwalliyar MG 500, haka kuma nau'in parenteral a ampoules (5 ml) na maganin 10%. Ana magance maganin maganin ta hanyar ciki, cikin intramuscularly, da parabulbarno (a cikin ophthalmology).

Yi la'akari da shahararrun magunguna - "Mildronate" 500, buɗe umarnin hukuma don amfani:

  • ana nuna magungunan don maganin angina pectoris da nau'ikan ischemia na na kullum da kuma cututtukan zuciya,
  • a cikin jiyya na rashin lafiyar zuciya na rashin aiki (rashin aiki mai rauni sosai),
  • tare da cardiomyopathies na asali daban-daban kuma tare da dystrophy na myocardial,
  • da aka nuna don cututtukan ischemic, cututtukan cututtukan kwakwalwa da kuma wahalar jini,
  • tare da gajiya da rage karfin aiki,
  • idan aka sami karin kaya, gami da wasanni,
  • a cikin lura da shan barasa (tare da cire alamun cirewa).

Wannan ita ce shaidar hukuma. Amma, a zahiri, ƙwayar tana iya ƙara ƙarfin hali, yana ƙaruwa da juriya ga damuwa, yana kunna tsarin juyayi na tsakiya, yana saurin dawo da jiki.

Wannan shine dalilin da ya sa likitoci da yawa suka fara ba da Mildronate ga kowane mai haƙuri, duka tare da cututtuka da don rigakafin.

Tabbas, wannan magani ya zama "panacea" ga waɗannan mutanen da ke da shakku, damuwa da hypochondria.

Sun yi imanin cewa idan ziyarar likitan ba ta ƙare da takardar magani ba, to ziyarar ba ta yi nasara ba, kuma likita ba shi da kyau. Mildronat ya girmama wannan yanayin.

Hankali! Yana da mahimmanci a fahimci cewa tare da dukkan "ƙari" a ko'ina cikin shaidar yana cewa: "ana amfani da miyagun ƙwayoyi a cikin maganin rikicewar cuta."Wannan yana nufin cewa daban-daban Mildronate ba zai iya ba, kuma bai kamata ba, cire ischemia myocardial, ko yin daidai a cikin sauran yanayi. Yana taimaka kawai don murmurewa da sauri.

Yaya ake amfani da miyagun ƙwayoyi?

Mildronate na iya samun sakamako mai ban sha'awa, har ma ya haifar da tashin hankali. Sabili da haka, waɗanda suke amfani dashi da farko, an bada shawarar kar su ɗauka daga baya fiye da 17.00 (idan an shirya bacci na al'ada da dare), amma zai fi kyau iyakance shi zuwa liyafar da safe. Akwai hanyoyin da yawa daban-daban na shan magani, gwargwadon ganewar asali:

  • Myocardial infarction da siffofin cututtukan zuciya na jijiyoyin zuciya suna buƙatar zuwa 1000 MG kowace rana, har zuwa watanni 1.5. Liyafar liyafar
  • Tare da dystrophies na myocardial da cardiomyopathies, 500 MG sau ɗaya ya isa, don kwanaki 10-14,
  • A cikin mummunan haɗarin cerebrovascular na yanayin ischemic (shanyewar jiki, hare-hare na ischemic na yau da kullun), ana gudanar da maganin a cikin ciki, alal misali, a hade tare da glucose, insulin da potassium chloride. Bayan hanya ta injections, ana sanya 1000 mg kowace rana da safe, ko 500 MG na kwalliyar Mildronate (safe da yamma) na tsawon watanni 1 zuwa 2.

Yin amfani da allurar Mildronate kuma an nuna shi azaman bolus ɗin cikin ciki. Ya kamata a tuna cewa ampoule guda ɗaya a cikin 5 ml yayi daidai da "babban" kwalliya a cikin 500 MG na miyagun ƙwayoyi, tunda abun ciki na meldonium shine 100 MG a cikin 1 ml na bayani.

  • Game da haɗari na ƙwayar cuta na ƙwayar cuta (ƙwayar cuta na atherosclerosis, ischemia na kullum), ana nuna magungunan don 500 MG sau ɗaya a rana, kuma tsawon lokaci - har zuwa watanni 2,
  • Ana ba da izinin shigar da 'yan wasa, kazalika da daidaikun mutane waɗanda aka fallasa su, ko kuma suka sami gagarumar ƙwaƙwalwa ta jiki a cikin sashi na 500 zuwa 1000 a kowace rana. Adadin shigowa daga makonni biyu zuwa uku,
  • A matsayin ɓangare na ƙwaƙƙwaran farfaɗar cututtukan cire barasa, ana nuna magungunan a cikin babban kashi - har zuwa 2000 MG kowace rana, an kasu kashi 4. Hanyar magani takaice - a kan matsakaici - 7 days.

Mutane da yawa suna tambaya - wanne yafi tasiri: shan allunan Mildronate, ko allura? Don amsar tambaya daidai, kuna buƙatar komawa zuwa kan magunguna da magungunan ƙwayoyi. An sani cewa mafi girman maida hankali ga jini plasma na faruwa 1 zuwa 2 sa'o'i bayan fitowar.

Dole ne kwayoyi su ratsa cikin hanta don kunnawa. Akasin haka, an lalace a cikin hanta, juya zuwa metabolites 3 zuwa 6 hours bayan shigowa.

Sabili da haka, yana da kyau a yi amfani da tsari mai injectable, tunda a wannan yanayin farkon sashi ta hanta an cire shi (bayan sha maganin a cikin duodenum a cikin yanayin capsules).

Tabbas, don wannan dole ne duk yanayi da tabbataccen shaida.

Mildronate (meldonium) a cikin wasanni: gaskiya, tsarin aikin, yadda za a karɓa kuma yana da ƙimar?

Tarihin mai laushi (meldonium) a cikin wasanni ya fara da sanannen ɗan wasan Tennis na Rasha Maria Sharapova. A shekara ta 2016, ta zama tauraruwar abin kunya, bayan kyakkyawan gwajin doping a gasar Australia Open.

Dalilin ba magungunan anabolic steroids bane, erythropoietin ko hormones, amma magani ne na maganin kadara, ga mamakin ba Sharapova kawai ba, har ma daukacin al'ummomin duniya har ma da 'yan wasa wadanda ke da kujera a kan harhada magunguna.

A cikin wannan labarin za mu bincika bayanai game da ilimin tauraron dan adam, gano menene dalilin aikin likitancinsa, tsarin aikin sa, da kuma wasu sakamako masu illa.

Gaskiya game da Mildronate (Meldonium)

  • Meldonium yana haɓaka kamfanin magunguna na Latvian
  • Meldonium mai hana iskar shaka mai kitse (yana hana kone su)
  • Hukumar Kula da Magunguna ta Duniya (WADA) ta haramta amfani da shi wurin motsa jiki.
  • Babban abin nuni ga yin amfani da maganin dan karatoci a magani shine maganin matsalolin zuciya, amma jerin abubuwan da ke nuna alamun suna da fadi sosai.
  • An haramta Meldonium don amfani (ba da lasisi ba) a Amurka, an yarda da shi a Rasha da wasu ƙasashe na tsohuwar kungiyar USSR
  • Sojojin Soviet sun yi amfani da maganin a lokacin yaƙin Afghanistan.

Menene meldonium (softronate)?

Meldonium ya haɓaka ta kamfanin kamfanin magunguna na Latvian Grendiks.

Ofaya daga cikin magunguna na farko don Mildronate shine haɓaka takin gargajiya (yawan maniyyi) a cikin aladu na maza da wasu dabbobi na gida. Bayan haka, an faɗaɗa ikon zuwa 2.

  • Sayar da maganin ya kasance kudin Tarayyar Turai miliyan 56 a shekara ta 2013, wanda ya sanya Grendiks ya zama babban dillalai a kasuwar magunguna ta Latvian.
  • Daga 1979 zuwa 1989, Mildronat ya ƙaddamar da babban "gwaji" akan sojan Rasha: an aika shi zuwa adadi mai yawa zuwa Afghanistan daga 1979 zuwa 1989.
  • Me yasa?
  • A cewar mai gabatarwa Ivan Calvins, tasirin meldonium shine inganta samar da iskar oxygen ga jiki.
  • Sojojin sun dauki meldonium yayin da suke cikin tsaunukan Afghanistan, lokacin da ya zama dole su dauki kayan aiki masu karfi: magani ya inganta juriya a yanayin iska mai santsi.

A yau, Mildronate magani ne wanda aka yi amfani da shi a Gabashin Turai da Asia ta Tsakiya (kasashen tsohuwar Soviet Union) don kula da yanayin likita da yawa, amma sama da duka cututtukan zuciya. A Amurka da wasu ƙasashe da yawa, an haramta.

Baya ga amfani da likita, ana amfani da meldonium sosai a cikin wasanni azaman wakilin doping wanda ke inganta aikin yi.

Tun daga farkon shekarar 2016, lokacin da Maria Sharapova ta kawo shi babban suna, 'yan wasa da yawa daga kasashe daban-daban (ciki har da Amurka, Rasha da kasashen Turai) WADA ne aka ba su sunayen ta don amfani da su.

Meldonium magani ne wanda manufar sa ta farko shine ƙara haɓaka aladu a aladu. A yau ana amfani dashi sosai don magance cututtukan zuciya.

Me yasa aka sanya Mildronate a magani?

A cikin magani, an wajabta Mildronate ga marasa lafiya waɗanda ke fama da wahalar jini zuwa wasu sassan jiki, musamman, tare da matsalolin zuciya da cututtukan jijiyoyin zuciya (wanda ke ciyar da zuciya da kanta), don maganin angina da ciwon zuciya.

Nazarin ilimin kimiyya ya tabbatar da ingancinsa a cikin magance cututtukan zuciya na zuciya 4 da bugun jini 5.

A wasu ƙasashe, ciki har da Rasha, Latvia, Ukraine, Georgia, Kazakhstan, Azerbaijan, Belarus, Uzbekistan, Moldova, da Kyrgyzstan, likitoci suna ba da izinin sauƙaƙe don inganta samar da jini ga kwakwalwa 6.

An nuna cewa yana inganta yanayi kuma yana haɓaka aikin motsa jiki, yana kawar da danshi da tashin zuciya 8.

Hakanan meldonium yana sauƙaƙe alamun bayyanuwa bayan shan giya.

Sauran alamomi don amfanin Mildronate 6:

  • ciwon ciki
  • raunin ido
  • cututtukan huhu da huhun hanji.

Idan ka karanta umarnin a hankali game da amfani da na'urar motsa jiki, za mu sami irin waɗannan maganganun “suna inganta aikin jiki da aikin tunani”, kodayake sashin "ba zai shafi aikin wasanni ba" kuma za a kasance a ciki.

Akwai bambanci, kamar yadda a bayyane yake cewa duk abin da ke inganta samar da jini, yana inganta wasan motsa jiki. Ayyukan da yawa na shirye-shiryen doping ya dogara da wannan ka'idodin.

Bayanin WADA na dalilin ƙara meldonium a cikin jerin magungunan hana yin allurar rigakafin, an mayar da hankali ne ga wannan kadara: "Meldonium yana ƙara yawan motsa jiki ta hanyar samar da oxygen zuwa tsarin jijiyoyin jini da tsokoki."

A cikin magani, an wajabta Mildronate don inganta wurare dabam dabam na jini zuwa ga gabobi daban-daban, gami da zuciya da kwakwalwa, da kuma rage alamun bayyanar buguwa bayan maye.

Mildronate (Meldonium) a cikin wasanni

Fitaccen dan wasan Mildronate a wasanni an kawo shi ne ta 'yar wasan Tennis ta Rasha, Maria Sharapova, wacce ba ta ba da izinin doping a watan Maris na 2016 ba, watanni uku bayan WADA 1 ta fitar da jerin sunayen.

Ta yarda cewa ta yi amfani da maganin tsawon shekaru 10 kamar yadda likitan ya umurce ta. Duba sake duba kwalliyar likitanci game da amfani da meldonium Sharapova.

  • Nan da nan bayan wannan fitowar, tallace-tallace na Mildronate sun girma sau da yawa.
  • Kusan lokaci guda tare da dakatarwar Sharapova, WADA ta karbi lambar adon Rasha Ekaterina Bobrova kuma a wannan shekarar, gwarzon duniya a cikin 1,500 m na gudu Abeba Aregawi, wanda ya lashe tseren Tokyo a 2015 Endeshaw Negesse.
  • Masu ba da lamuni na 13 na wasannin Turai a Baku a cikin 2015 sun kuma nuna kyakkyawan gwaji don amfani da meldonium, kuma masana sun ba da shawarar cewa yayin gudanar da su, kusan 470 duk mahalarta sun ɗauki maganin 17.
  • Tun daga wannan lokacin, an kara fadada yanayin kasa, kuma 'yan wasa daga Rasha, Habasha, Sweden, Jamus da Ukraine sun sha kama a lokuta daban-daban ta amfani da meldonium.

Da zato 17% na 'yan wasan Rasha suna amfani da meldonium kuma kawai 2% a wasu ƙasashe. Idan lambar tayi daidai, to wannan ya tabbatar da ingancinsa.

Rushewar doping kwanan nan da kuma hana shiga DUK na kungiyar Rasha a wasannin Olympics kai tsaye yana nuna cewa masana'antar doping ta Rasha, wacce ke goyan bayan wasannin kwararru, tana daya daga cikin karfi kuma mafi daukaka a duniya.

Mildronate ta samu karbuwa sosai a wasannin da aka yi godiya ga sunan 'yar wasan Tennis ta Rasha Maria Sharapova: bayan fitarta, tallace-tallacen magungunan sun karu sau da yawa.

Dangane da WADA rarrabewa, meldonium yana cikin rukuni na masu gyara metabolism, ban da insulin 7.

Idan kuna ganin yana da mahimmanci muyi - goyi bayan aikinmu!

Don tunani. An haɗa abu a cikin takardar doping idan:

  • yana haɓaka wasan motsa jiki,
  • yana haifar da barazana ga lafiyar 'yan wasa,
  • ya keta ruhun gasa.

Ma'anar hujja ta farko a bayyane take: mai tsere mai shan irin waɗannan ƙwayoyi yana samun fa'ida akan wasu. Bayani na biyu ya shafi kusan kowane magani na likita, tunda dukansu suna da tasirin sakamako masu illa. Amma ma'anar ta ukun ita ce mafi tsananin zafi kuma yana baka damar "ban" gaba ɗaya kowane abu.

"Meldonium ya nuna haɓaka athletesan wasa masu haƙuri, post-motsa jiki dawo da kudaden, kariya daga danniya da kuma juyayi tsarin aiki. ”

Babban jigon amfanin meldonium a wasanni wani abu ne kamar haka:

  • yana ƙaruwa gabaɗaya aikin jiki,
  • yana inganta samar da iskar oxygen zuwa tsokoki,
  • yana hanzarta fitar da ƙwayar jijiya (wannan yana da mahimmanci don saurin amsawa),
  • taimaka a cikin yaki da danniya shafi tunanin mutum yayin gasa,
  • yana inganta wadatar zuciya da kwakwalwa kwakwalwa tare da glucose = makamashi,
  • yana hanzarta kawar da kayan lalata.

Tasirin Mildronate, wanda yake da mahimmanci ga 'yan wasa, shine inganta samar da iskar oxygen da glucose ga tsokoki, ƙara yawan amsawar da tasirin tashin hankali

Hanyar aikin meldonium

  • Sakamakon warkewa na meldonium shine tarewa aikin carnitine, wanda ke cikin haɓakar mai na mai (ƙona su don makamashi), don amfanin farko na glucose 3.
  • Lokacin aiwatar da motsa jiki na iska (wanda ke cin yawancin oxygen), L-carnitine yana da tasiri ga aikin zuciya, yana sa hadawar iskar gas mai inganci ga kuzari: kusan kashi 80% na kuzarin an samar dashi ta amfani da wannan inji 10.
  • Koyaya, a cikin jihar da babu isasshen oxygen a cikin sel, abubuwa masu guba suna tarawa - samfuran fatima mai ƙanshi.
  • Abin da ke sa meldonium: yana hana tsarin hadawar kitse mai kazari ta hanyar carnitine (rage maida hankali a cikin sel) da kuma kunna amfani da sinadarin glucose, wanda shine farkon kuma mafi ingancin tushen kuzari a jiki, tunda yana bukatar karancin iskar oxygen 11-13 don magance shi.
  • Haka kuma, Mildronate kai tsaye yana motsa glycolysis, wanda ke kara haɓaka ƙarfin ƙarfin ɗan wasa 14.

Shin yana da ma'anar ɗaukar matsin lamba (meldonium) a cikin gina jiki?

  1. Meldonium ya shahara musamman a wasannin motsa jiki, alal misali, tsakanin dillalai da masu gudu a cikin su wanda saurin gudu da amsawa suna da mahimmanci.
  2. Dangane da amfani da matsin lamba kan gyaran jiki da fadada karfin iko, sabanin mashahurin imani, shi KADA KA shafi kai tsaye ci gaban tsoka.
  3. A cikin wasanni motsa jiki ana amfani dashi. don sauwaka alamun bayyanar da damuwa, wanda yake da dacewa kawai ga foran wasan kwararru.

Karanta mana a yanar gizo

Wanne ya fi kyau: rage nauyin ko ƙara wani kwaya a cikin maganin ƙirar maganin ku - ku yanke shawara.

Mildronate a cikin ginin jikin mutum ba shi da tasiri kai tsaye ga ci gaban tsoka, ana amfani dashi don magance alamun rashin gamsuwa

Yadda ake ɗaukar Mildronate don 'yan wasa: umarni

Alamar daukar meldonium a cikin wasanni wasanni ne na yau da kullun.

A cikin nazarin ilimin kimiyya wanda ke nuna tasirin sakamako mai laushi ga 'yan wasa masu ƙwararru, ana amfani da allurai na 0.25-1 g sau biyu a rana don makonni 2-3 na lokacin horo, kwanaki 10-14 kafin gasar.

Lokacin karbar sosai daidaitaccen sashi yana da mahimmanci. Ana kirga kashi na yau da kullun akan 15-20 mg ta kilogram na nauyin jiki.

An yarda da Meldonium a cikin wasanni (da gina jiki) Lokaci 1 a rana minti 30 kafin horo.

Har yaushe zan iya ɗaukar Mildronate ba tare da hutu ba?

Tsawon lokacin daga aji shida ne zuwa watanni 3. Bayan wannan, jikin yana inganta jaraba ga miyagun ƙwayoyi, yana asarar tasiri. Bayan hutu na makonni 4, an sake dawo da mai saukin kamuwa.

Ana iya ɗaukar Meldonium a cikin nau'i biyu: allunan da injections. A cikin nau'ikan allunan, kashi na yau da kullun kada ya wuce gram 2. Inje shine kamar sau biyu.

Wani lokaci ana shawarar Mildronate tare da L-carnitine da Riboxin. A magana ta farko, akwai rashin inganci, tunda tsarin aikin sirinda shine toshe aikin carnitine.

Ana ɗaukar Meldonium a cikin wasanni da gina jiki a cikin adadin 15-20 a kowace nauyin nauyin jiki 1 lokaci kafin horo

Har yaushe za a fitar da meldonium?

  • Babu amsa mai ban haushi ga tambayar game da lokacin kawar da meldonium daga jiki, tunda masana kimiyya basuyi nazarin shi ba.
  • Wasu majiyoyi suna ba da rahoton cewa matsakaicin lokacin cirewa shine 24 hours tare da kashi daya, idan ana shanta akai-akai, to ganowa cikin jini yana yiwuwa ko bayan hakan watanni da yawa bayan daina amfani.
  • Wasu masana sun ce cikakkiyar kawar da abubuwa masu sauki daga jiki na faruwa a cikin kwanaki 100-120.

Jimlar lokacin kawar da meldonium daga jiki zai iya kai watanni 3-4 tare da amfani na yau da kullun

Mildronate: sakamako masu illa

Binciken data kasance yana ba da shawara babu mummunan sakamako masu illa a cikin meldonium.

Koyaya, bisa ga ra'ayoyin masana ilimin likitanci, likitoci sunyi la'akari da wannan batun ba a fahimta sosai.

Ana nuna alamun illa na yau da kullun a cikin umarnin don amfani da mara lafiyar:

  • rashin lafiyan mutum
  • tachycardia (hawan jini a zuciya),
  • narkewa a cikin abinci.

Bayanna

Mildronate samfuri ne na masana'antar doping na gida, wanda 'yan wasa daga ko'ina cikin duniya ke son gwadawa (godiya ga Mariya Sharapova saboda wannan).

Rarrabawa da amfani da 'yan wasan Rasha ke amfani da shi yana nuna yuwuwar tasirinsa. Bayan 'yan karatun kimiyya sun tabbatar da amfani da meldonium a cikin wasanni na motsa jiki (gudu, tsere, kekuna) da tsaka-tsaki a cikin iko (ginin, motsa jiki).

An cire Mildronate daga jiki tsawon watanni kuma baya da mummunar illa.

Amfani da magani don lura da cututtukan zuciya

A cikin mutanen da ke da lalacewa na jijiyoyin jini, gazawar zuciya, ana amfani da maganin don inganta metabolism na sel tsoka. Tasirin ƙwaƙwalwar zuciya na Mildronate a cikin lura da cututtukan jijiyoyin zuciya da kuma sakamakon cututtukan zuciya ya ƙunshi tasirin:

  • toleara haƙuri da ƙwayar zuciya ga damuwa,
  • raguwa daga yankin necrosis,
  • inganta hawan jini a yankin da abin ya shafa,
  • raguwa a tsawon lokacin farfadowa.

A cikin marasa lafiya da ke fama da cututtukan zuciya na yau da kullun, ƙwayar ta sami damar rage yawan tashin hankalin angina. Hakanan, ƙwayar, kamar yadda aka nuna a cikin umarnin, yana ƙaruwa da ƙarfi na ƙanƙancewar ƙwayar zuciya da fitarwa na zuciya. Tare da amfani na yau da kullun, Mildronate yana rage jinkirin ƙarancin hanyoyin cututtukan da ke faruwa a cikin myocardium.

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