Menene saukad da methyl ethyl pyridinol na?

Alurar ta fito sarari, ba ta da launi ko tawaya mai haske.

1 ml
methylethylpyridinol hydrochloride10 MG

Fitowa: hydrochloric acid 0.1 M bayani - har zuwa pH 2.5-3.5, ruwa d / i - har zuwa 1 ml.

1 ml - gilashin ampoules (5) - fakitin bakin ciki (1) - fakitoci na kwali.
1 ml - gilashin ampoules (5) - fakitin bakin ciki (2) - fakitoci na kwali.
1 ml - gilashin ampoules (5) - fakitoci na kwali.
1 ml - gilashin ampoules (10) - fakitoci na kwali.

Aikin magunguna

Angioprotector, yana rage yiwuwar bango na jijiyoyin bugun gini, shine mai hana ayyukan tsoma baki, antihypoxant da antioxidant.

Yana rage dankowar jini da tarawar platelet, yana kara yawan sinadarin cyclic nucleotides (cAMP da cGMP) a cikin platelet da kwakwalwar kwakwalwa, yana da aikin fibrinolytic, yana rage yiwuwar bango na jijiyoyin bugun jini da kuma hadarin basur, yana inganta resorption din su. Yana faɗaɗa tasoshin jijiyoyin jini, a cikin tsawan lokaci na infitar ƙarfin ƙwaƙwalwa na ƙuntata girman girman ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwar ƙwayar cuta, yana inganta daidaituwa na zuciya da aikin tsarin sa. Tare da haɓakar jini yana da sakamako mai illa. A cikin mummunan ischemic cuta na cerebral wurare dabam dabam yana rage tsananin bayyanar cututtuka na jijiyoyin jini, yana ƙaruwa da juriya tsakanin tsoka da ischemia.

Yana da kyan gani na kariya, yana kare retina daga illolin tasirin haske mai-ƙarfi, yana inganta yanayin zubar jini, inganta microcirculation na ido.

Alamar magunguna

A matsayin wani ɓangare na hadaddun farji: sakamakon hatsarin cerebrovascular of ischemic and hemorrhagic nature, kai rauni, postoperative period of epi- and subdural hematomas, myocardial infarction, anti of reerfusion syndrome, rashin bacci angina pectoris.

Subconjunctival da bashin jini na ciki, angioretinopathy (ciki har da masu ciwon sukari), chorioretinal dystrophy (gami da atherosclerotic asali), dystrophic keratitis, kashin baya na jijiyoyin bugun jini, rikicewar cututtukan mahaifa, kariya daga kasala (lokacin saka tabarau ta ido) da kuma retina na ido haske mai ƙarfi (Laser da kunar rana a jiki, tare da laser-coagulation), rauni, kumburi da ƙonewar cornea, cataract (gami da rigakafin cikin mutane sama da 40), tiyata ta ido, yanayin bayan tiyata don r laucoma tare da chocho choachment.

Lambobin ICD-10
Lambar ICD-10Nuna
F07Halin mutum da rikicewar halaye saboda rashin lafiya, lalacewa, ko lalatawar kwakwalwa
F07.2Ciwo bayan-rikicewar cuta
H20.2Lens iridocyclitis
H21.0Hyphema
H31.1Ciwan Choroidal
H31.2Magungunan gado na choroid
H34Kasancewa na Jijiyoyin bugun ciki
H35.6Kwakwalwar koda
H36.0Rashin maganin ciwon sukari
H52.1Myopia
I20.0Angina mai tsauri
I21Babban myocardial infarction
I61Cutar ciki na ciki (nau'in basur na nakasar ciki)
I63Cerbral infarction
I69Sakamakon cututtukan cerebrovascular
T26Ronawa da sinadarai suna ƙone iyakance ga ido da adnexa

Sakawa lokacin

A cikin neurology da cardiology - iv drip (20-40 saukad da / min), 20-30 ml na maganin 3% (600-900 mg) sau 1-3 a rana don kwanaki 5-15 (a baya ana amfani da maganin a cikin 200 ml na 0.9% maganin NaCl ko bayani 5% na dextrose). Tsawon lokacin jiyya ya dogara da cutar. Bayan haka, suna canzawa zuwa gudanarwa na wucin gadi - 3-5 ml na bayani na 3% sau 2-3 a rana don kwanaki 10-30.

A cikin maganin ophthalmology - subconjunctival ko parabulbar, lokaci 1 kowace rana ko kowace rana. Subconjunctival - 0.2-0.5 ml na 1% bayani (2-5 mg), parabulbar - 0.5-1 ml na 1% bayani (5-1 mg). Tsawon lokacin jiyya shine kwanaki 10-30, yana yiwuwa a maimaita karatun sau 2-3 a shekara.

Idan ya cancanta, retrobulbar a cikin 0.5-1 ml na 1% bayani 1 lokaci kowace rana don kwanaki 10-15.

Don kare retina yayin coagulation na laser (ciki har da iyakance da lalata coagulation na ciwace-ciwace) - parabulbar ko retrobulbar 0.5-1 ml na 1% bayani 24 hours da awa 1 kafin coagulation, to a cikin allurai guda (0.5 ml kowace) 1% mafita) 1 lokaci a rana don kwanaki 2-10.

Sunan kasuwanci

A cikin cibiyar sadarwar rarraba, ana kiran saukadden idanu Emoxipin, tare da babban sinadaran aiki methylethylpyridinol (methylethylpiridinol). Hankalinsa a cikin bayani shine 1%, i.e., 1 ml na miyagun ƙwayoyi ya ƙunshi 10 MG na babban abu.

Ana samun zubar ruwan ido a cikin filastik, sanye take da farar ruwa, kwalabe cike da ruwa mai tsafta, mara launi. Volumearar kowane 5 shine ml 5 ko 10. Ana cika kwalayen cikin akwatunan kwali tare da cikakkun bayanan umarnin da aka haɗe.

Analog na wadannan saukad da shine Emoxy-Optic.

Hakanan ana samun Methylethylpyridinol a cikin ampoules 1 ml. Hakanan ana amfani da wannan nau'in magungunan don magance cututtukan ido kuma ana iya sarrafa shi a karkashin abu (ƙananan gefen ido) ko kai tsaye zuwa orbit na ido (ƙananan rabin ƙwallon ido). Ana amfani da waɗannan hanyoyin na maganin magunguna a cikin coagulation na laser.

Dangane da umarnin, ana iya adana ganyen Emoxipin sama da kasa fiye da + 25 ° C tsawon shekaru 2, kuma bayan buɗe shi - ba fiye da kwanaki 30 ba. Ya kamata a kiyaye wurin ajiya daga hasken rana kai tsaye kuma a nesa da kananan yara.

Umarnin don amfani: alamomi da contraindications

Ana amfani da fuka-fukan ido Emoksipin don magance cututtukan idanu da yawa, amfanin su kuma yana yiwuwa ga dalilai na prophylactic:

  • Ciwon mara na Angola - wani rikitarwa na pathology tare da dogon tafiya na cutar, aka bayyana a cikin raunuka na jini,
  • Glaucoma - raunin gani tare da na lokaci zuwa lokaci ko yawan karuwa a cikin jijiya,
  • Myopia - myopia, lokacin da hasken rana yake shiga cikin ido yana mai da hankali a wani lokaci ba tare da ya isa cikin satin ba. Sakamakon haka, mutum ba ya bambanta abubuwa sama da nisa,
  • Hypermetropia - farsightedness, kishiyar myopia. Mai haƙuri yana iya gani sosai a cikin nesa, kuma a kusa da abubuwa suna fitar da fitila,
  • Yana ƙone idanu - lalacewar kwasfa na waje sakamakon fashewar sinadarai, high t, ultraviolet radiation, vapors.

Karanta ƙari game da cutar ta glaucoma anan.

Methylethylpyridinol shine ingantacciyar kayan aiki a cikin lura da tafiyar matakai masu kumburi a cikin membranes na waje, tare da bashin bayan-traumatic, da rikitarwa na conjunctivitis.

Daidaitaccen tsarin amfani da shi ya kunshi koyarwa a cikin kowane ido 1 sauke sau 2-3 a rana. Matsakaicin tsawon lokacin kulawa shine kwana 3-10. Koyaya, kamar yadda likita ya umarta, za'a iya tsawaita hanya zuwa wata 1. Inganta tasirin magani ana samunshi ta hanyar bin fewan ka'idoji kaɗan:

  • A wanke hannun sosai da sabulu kafin da bayan aikin,
  • Kafin amfani da dropper, bincika ka gani ko akwai wasu abubuwan ƙonewa a ƙarshen da zasu iya lalata ido,
  • Lokacin da kake farawa, kar a taba mai dattin din a saman idanun,
  • Bayan hanyar, rufe gashin ido, kuma cire duk wani danshi wanda ya bayyana tare da kyallen mai bakararre,
  • Cire ruwan tabarau na hulɗa kafin farawa a cikin mintina 15. , da sutturar da ba ta wuce mintuna 15 ba. bayan hanya.

Kuna iya karanta rubutun don binciken idanu a nan.

Yayin aikin jiyya, hangen nesa zai iya yin fuska, saboda haka, mutanen da ke gudanar da ayyukan da ke bukatar karin hankali ya kamata su huta.

Contraindications

Jerin contraindications na Emoxipin ya ƙunshi mafi ƙarancin abubuwa, tare da duk abubuwa masu alaƙa da abubuwan da aka saba samu a cikin kusan kowane magani.

An hana amfani da idanun methylethylpyridinol gaban halaye masu zuwa:

  • Hypersensitivity ga aiki abu da sauran aka gyara,
  • Shekarun haƙuri ba su wuce shekara 18 ba
  • Lokacin haihuwar da ciyar da yaron.

Ya kamata a kula da kulawa ta musamman a cikin marasa lafiya tare da halayen halayen halayen rashin lafiyan, musamman a farkon jiyya. Idan akwai wani rashin jin daɗi wanda baya ɓacewa akan hanyoyin da yawa, ya kamata a dakatar da magani kuma ya kamata a sami ƙarin shawarar likita.

A lokacin daukar ciki

Lokacin haila (lokacin haihuwa) - daya daga cikin masu daukar nauyin rayuwar kowace mace. Duk wani magani ba a ke so ba yayin daukar ciki, saboda a koyaushe akwai kankanin haɗarin yin mummunar illa ga tayin. Wasu abubuwa har ma suna da ikon shiga cikin mahaifa.

Tabbas, lokacin amfani da saukad da idanu, ƙwaƙwalwar tsari yana faruwa cikin adadi kaɗan. Koyaya, methyl ethyl pyridinol abu ne mai ƙarfi mai ƙarfi wanda ke shafar yawancin matakan rayuwa a cikin jiki.

Haramcin amfani da miyagun ƙwayoyi ya samo asali ne sakamakon rashin ingantaccen bayanai kan sakamakon amfani da shi, tunda, a zahiri, ba a gudanar da gwaje-gwaje a kan mata masu juna biyu. Sabili da haka, tunda magani ne takardar sayan magani, amfaninsa don magani yana cikin shawarar likita.

Inalwaƙwalwar ƙwayar cuta na fata - magani tare da magungunan jama'a da magunguna an bayyana su a wannan labarin.

Yara kanana

Dangane da kula da yara, umarnin a bayyane yake yana hana shekaru zuwa shekaru 18 - kafin hakan, ba a ba da shawarar kula da yara ba. Koyaya, wasu masana'antun har yanzu suna nufin gaskiyar cewa wannan hani kuma an samo asali ne daga rashin ingantaccen sakamako game da amfani da miyagun ƙwayoyi.

Kara karantawa game da faduwar ido Dexamethasone a mahadar.

A aikace, likitocin dabbobi sukan bada shawarar Emoxipine har ma ga kananan yara, tunda magungunan yara masu tasiri don wasu cututtukan idanu kawai ba su wanzu.

Matsaloli da ka iya haifar da kwayoyi

Nazarin masu haƙuri sun nuna cewa an yarda da miyagun ƙwayoyi gaba ɗaya. A cikin halayen da ba a sani ba, jin dadi mara dadi a cikin yanayin halayen halayen mai yiwuwa ne: ƙona, itching, jan launi, lacrimation.

Game da amfani da haɗin gwiwa tare da wasu kwayoyi, ana bada shawara don amfani da Methylethylpyridinol na ƙarshe, bayan aƙalla minti 15. bayan amfani da magani na ƙarshe.

Game da saukad da idanu don Tsiprolet an rubuta a cikin labarin.

Kamar yadda analogues na miyagun ƙwayoyi, Emoxy-optic, Emoxipin-AKOS, Emoxibel za'a iya amfani dashi.

Wannan miyagun ƙwayoyi magani ne mai matuƙar tasiri wanda zai iya yin tasiri ga yawancin hanyoyin metabolism a cikin kyallen ido. Sabili da haka, amfani da shi don dalilai na warkewa da kuma dalilai na prophylactic za a iya barata a gaban abubuwan da yawa, tare da barazanar ci gaban su.

Duk da gaskiyar cewa magungunan magani hanya ce ta bayyanuwa gabaɗaya, amfaninsa ya kamata ya zama baratacce kuma ana aiwatar dashi ne kawai a ƙarƙashin kulawar likitan likitan ido.

Hakanan karanta game da kwayoyi irin su ciprofloxacin saukad da kayan.

Formaddamar da tsari da abun da ke ciki

Form sashi - allura: bayyananne, mara launi ko ruwa mai launin rawaya mai haske, 1 ml kowane a cikin ampoules na tsaka mai tsami gilashin ko gilashin tare da rukunin jigilar hydrolysis na HGA1, a cikin kwali na fakiti 5 ko 10 ampoules cikakke tare da ampoule scarifier (lokacin ɗaukar ampoules tare da ba a saka mai ɗinki ba tare da zobe ko aya mai fashewa) ko fakiti na 1-2 na murfin 5 ampoules da umarnin don amfani da Methylethylpyridinol, marufi don asibitoci - a cikin kwali na kwali na 4, 5, 10, 50 ko 100 kwano-kwano fakitoci to 5 vials.

Abun ciki na 1 ml na bayani:

  • abu mai aiki: methylethylpyridinol (a cikin nau'i na hydrochloride) - 10 MG,
  • abubuwan taimako: 0.1 M hydrochloric acid bayani, ruwa don allura.

Pharmacodynamics

Methylethylpyridinol antioxidant ne, mai hana ayyukan tsattsauran ra'ayi ne.

Yana da tasiri mai amfani akan tsarin coagulation na jini: yana rage danko na jini, yana tsawanta lokacin coagulation, kuma yana hana tarawar platelet. Yana kwantar da membranes na sel jini da sel jijiyoyin jini, ƙara juriya da jini jini to haemolysis da na inji rauni.

Yana haɓaka abubuwan da ke cikin cyclic nucleotides a cikin platelet (cyclic adenosine monophosphate da cyclic guanosine monophosphate), yana rage lalacewar bango na jijiyoyin bugun jini, yana inganta resorption na basur, kuma yana da aikin fibrinolytic.

Inganta microcirculation a cikin kyallen ido, gami da tasoshin retina. Yana da ma'anar retinoprotective, yana kare retina daga lalata abubuwan haske mai ƙarfi.

Alamu don amfani

Ana amfani da Methylethylpyridinol a matsayin wani ɓangare na hadaddun farke don cututtukan / yanayin:

  • dystrophic cututtuka na cornea,
  • Cutar kwalliyar ciki da tsokar jini wanda yake da asali daban-daban,
  • tsakiya da kuma na gefe choystretinal dystrophy,
  • ciwon zuciya (har da masu ciwon sukari),
  • angiosclerotic macular degeneration (bushe bushe),
  • thrombosis na tsakiyar jijiya na retina da rassanta,
  • rikice-rikice na daga myopia,
  • Digiri na biyu na ƙonewa da raunin jiki,
  • ware chocho a cikin bayan aikin tiyata bayan tiyata na glaucoma,
  • lalacewar ido tare da haske mai tsananin ƙarfi (radar laser yayin coagulation laser) - magani da rigakafin.

Methylethylpyridinol, umarnin don amfani: hanyar da sashi

Ana sarrafa maganin allurar Methylethylpyridinol parabulbarno (s / b) ko kuma subconjunctival (s / c). Ana amfani da miyagun ƙwayoyi a matsayin wani ɓangare na tasirin magani.

Nagari hanyoyin bada shawara:

  • cututtukan dystrophic na cornea: s / c 0.5 ml sau ɗaya a rana a cikin kwanakin 10-30,
  • Cutar kwalliyar ciki da kwatancen jini na tsokoki daban-daban: s / c ko p / b 0.5 ml sau ɗaya a rana don kwanaki 10-15,
  • tsakiya da na waje choystretinal dystrophy, bushe nau'i na angiosclerotic macular degeneration: 0.5 ml p / b sau ɗaya a rana don kwanaki 10-15,
  • thrombosis na tsakiyar jijiya na retina da rassanta: n / a 0.5 ml sau ɗaya a rana a cikin tafiyar kwanaki 10-15,
  • rikitarwa myopia: p / b 0.5 ml sau ɗaya a rana don kwanaki 10-30, idan ya cancanta sau 2-3 a shekara, maimaita karatun,
  • raunin da konewa na cornea na digiri na biyu: p / b 0.5 ml 1 sau ɗaya kowace rana don kwanaki 10-15,
  • detchment na choroid a cikin bayan aikin asibiti bayan tiyata na glaucoma: s / c ko p / b, 0.5-1 ml kowane sauran rana, hanya ta lura ta ƙunshi injections 10,
  • Kariyar retinal yayin coagulation na laser (ciki har da iyakancewa da ɓarna coagulation na ciwace-ciwace): 0.5-1 ml p / b 24 sa'o'i da 1 h kafin coagulation, sannan 0.5 ml sau ɗaya a kowace rana na tsawon kwanaki 2-10.

Side effects

  • halayen gida: ƙonewa, zafi, hyperemia, itching, compaction na paraorbital kyallen takarda (baya buƙatar kulawa ta musamman, yana warware kansa),
  • halayen rashin lafiyan: itching, peeling na fata, edema, hyperemia,
  • daga tsarin juyayi: bacci, tashin hankali na ɗan lokaci,
  • daga tsarin zuciya: fatar fata, hauhawar jini.

Hulɗa da ƙwayoyi

Methyl ethyl pyridinol bai dace da magunguna ba, saboda haka haramun ne a haxa shi a cikin sirinji guda tare da wasu kwayoyi.

Misalin Methylethylpyridinol sune: Vixipin, Cardioxypine, Methylethylpyridinol-Eskom, Emoxy-optician, Emoxibel, Emoxipin, Emoxipin-AKOS, da sauransu.

Neman bayanai game da Methylethylpyridinol

Nazarin game da methylethylpyridinol kaɗan, amma tabbatacce. Magungunan sun nuna inganci sosai, ba shi da tsada.Koyaya, bisa ga marasa lafiya, ya fi dacewa don amfani da kwayoyi tare da abu ɗaya mai aiki a cikin hanyar saukad da idanu.

Methylethylpyridinol galibi ana amfani dashi duka don cututtukan ophthalmological daban-daban, da kuma don rikicewar jijiyoyin jini da cututtukan zuciya.

Methylethylpyridinol: farashin a cikin kantin magani na kan layi

Methylethylpyridinol allurar 10 MG / ml don kwaya 1 ml 10.

Methylethylpyridinol bayani d / in. 10 mg / ml amp. 1ml №10 ELLARA

Ilimi: Jami'ar Kiwon lafiya ta jihar Rostov, kwararrun "General Medicine".

Bayanai game da miyagun ƙwayoyi an samar da su duka, an bayar da su don dalilai na bayanai kuma baya maye gurbin umarnin hukuma. Kai magani yana da haɗari ga lafiya!

Ya kasance hakan yana haɓaka jiki da oxygen. Koyaya, an rarraba wannan ra'ayin. Masana ilimin kimiyya sun tabbatar da cewa hayaniya, mutum yana sanya kwantar da hankali da haɓaka aikinsa.

Mutumin da yake da ilimi bashi da saukin kamuwa da cututtukan kwakwalwa. Aikin mai hankali yana bada gudummawa ga samuwar karin nama don rama marassa lafiya.

Cutar hanta ita ce mafi girman jikinmu. Matsakaicin nauyinta shine kilogiram 1.5.

Idan kun fada daga jaki, to, zaku sami damar juyar da wuyan ku fiye da wanda kuka faɗi daga doki. Kawai kada kuyi kokarin musun wannan magana.

Wani dan Australiya mai shekaru 74 James Harrison ya zama mai bayar da gudummawar jini kusan sau 1,000. Yana da nau'in jini wanda ba a taɓa gani ba, rigakafin cututtukan rigakafi waɗanda ke taimaka wa jarirai masu ƙarancin rashin wadatar rayuwa. Don haka, Ostiraliya ta sami kusan yara miliyan biyu.

An kirkiro firikwensin farko a karni na 19. Ya yi aiki a kan injin tururi kuma yana da niyyar kula da cutar mace.

Jinin ɗan adam "yana gudana" ta cikin jiragen ruwa a ƙarƙashin matsanancin matsin lamba, kuma idan an keta mutuncin sa, zai iya harba har zuwa mita 10.

Masana kimiyya daga Jami'ar Oxford sun gudanar da karatu da dama, a lokacin da suka kai ga matsayin cewa cin ganyayyaki na iya zama illa ga kwakwalwar dan Adam, saboda hakan yana haifar da raguwa a yawanta. Saboda haka, masana kimiyya sun bada shawarar kar a cire kifi da nama gaba daya daga abincin da suke ci.

A cikin 5% na marasa lafiya, maganin antidepressant clomipramine yana haifar da inzali.

A lokacin rayuwa, matsakaicin mutum ya samar da kasa da ruwa biyu na yau.

Yayin aiki, kwakwalwarmu tana amfani da adadin kuzari daidai da wutar fitila 10-watt. Don haka hoton gilashin haske sama da kanka a lokacin bayyanar tunani mai ban sha'awa ba ya da nisa da gaskiya.

Likitocin hakora sun bayyana ne kwanan nan. A cikin ƙarni na 19, aikin maikatar gashi ne na al'ada don fitar da hakoran da ke da lafiya.

Shahararren magungunan "Viagra" an samo asali ne don maganin hauhawar jini.

Yawancin mata suna iya samun ƙarin jin daɗi daga tunanin kyakkyawan jikinsu a cikin madubi fiye da jima'i. Don haka, mata ku yi ƙoƙari don jituwa.

Magunguna da yawa an fara tallata su azaman magunguna. Misali, a farko, an siyar da Heroin azaman maganin tari. Kuma likitoci sun ba da shawarar yin amfani da cocaine a matsayin maganin hana haihuwa da kuma hanyar wadatar da haƙuri.

Polyoxidonium yana nufin magungunan immunomodulatory. Yana aiki akan wasu sassan tsarin na rigakafi, ta haka yana ba da gudummawa ga haɓaka kwanciyar hankali na.

Pharmacokinetics

Volumearar watsawa - 5.2 lita. Cire rabin rayuwar shine mintina 18. Jimlar amincewa shine 0.2 l / min. Metabolized a cikin hanta. Kodan ya fice.

A wani ɓangare na hadaddun far:

  • Subconjunctival da jijiyoyin jini na jini na asali,
  • Cutarwar zuciya (har da masu ciwon sukari),
  • Tsakiya da kuma na mahaifa choystretinal dystrophy,
  • Thrombosis daga cikin jijiya na tsakiya da kuma rassan sa,
  • Hadarin cutar myopia
  • Angiosclerotic macular degeneration (bushe bushe),
  • Akewar choroid a cikin bayan aikin tiyata bayan tiyata na glaucoma,
  • Dystrophic cututtuka na cornea,
  • Raunin, ƙonewa ga cornea,
  • Jiyya da rigakafin raunuka na ido tare da hasken mai tsananin ƙarfi (hasken rana, radar laser yayin coagulation laser).

Sashi da gudanarwa

Ana amfani da miyagun ƙwayoyi a matsayin wani ɓangare na tasirin magani.

Tare da subconjunctival da cututtukan ƙwayar cuta na ciki-ciki na asalin asali - subconjunctival ko parabulbar 0.5 ml sau ɗaya a rana. Aikin magani shine kwanaki 10-15.

Tare da angioretinopathy (ciki har da masu ciwon sukari) - parabulbarno 0.5 ml sau 1 a rana. Aikin magani shine kwana 10.

Tare da dystrophy na tsakiya da na yanki, da kuma gurguwar macular antisclerotic (bushe bushe) - parabulbar 0.5 ml sau ɗaya a rana. Aikin magani shine kwanaki 10-15.

Tare da thrombosis daga cikin jijiya na tsakiya da rassa - parabulbarno 0.5 ml sau ɗaya a rana. Aikin magani shine kwanaki 10-15.

A cikin rikitarwa myopia - parabulbarno 0.5 ml sau ɗaya a rana. Aikin magani shine kwanaki 10-30, yana yiwuwa a maimaita karatun sau 2-3 a shekara.

Tare da lalata choroid a cikin marasa lafiya tare da glaucoma a cikin bayan aikin - parabulbar ko subconjunctival 0.5-1.0 ml sau ɗaya kowace kwana 2. Hanyar magani shine allura 10.

Don raunin rauni da ƙonewa na cornea na digiri na 2 - parabulbarno 0.5 ml sau ɗaya a rana. Hanyar magani shine allura 10-15.

Tare da cututtukan dystrophic na cornea - subconjunctival 0.5 ml sau ɗaya a rana. Aikin magani shine kwanaki 10-30.

Don kare retina yayin coagulation na laser (ciki har da iyakancewa da lalata coagulation na ciwace-ciwace), 0.5-1.0 ml na 1% bayani (5-10 mg) parabulbarly 24 hours da awa 1 kafin coagulation, to a cikin allurai guda ( 0.5 ml na 1% bayani) 1 lokaci a rana don kwanaki 2-10.

Yawan damuwa

Game da yawan abin sama da ya kamata, karuwa a cikin tsananin zafin cutar ya dogara da maganin yana yiwuwa.

Bayyanar cututtuka: haɓaka haɓakar jini, tashin hankali ko nutsuwa, ciwon kai, jin zafi a cikin zuciya, tashin zuciya, rashin jin daɗi a cikin yankin epigastric. Rashin rikicewar jini.

Jiyya: karɓar magani, maganin warkewa, babu takamammen maganin cutar kansa.

Umarni na musamman

Dole ne a gudanar da jiyya tare da methylethylpyridinol a ƙarƙashin ikon hawan jini da coagulation na jini.

Tasiri a kan ikon tuka motoci da aiki tare da kayan aiki

Tare da haɓakar nutsuwa, ya zama dole a guji tuki motoci da sauran hanyoyin motsawa, sannan kuma a mai da hankali yayin yin ayyukan haɗari waɗanda ke buƙatar haɓakar haɓaka da saurin halayen psychomotor.

Bayanin mai aiki mai aiki Methylethylpyridinol / Methylaethylpiridinolum.

Tsarin tsari C8H11NO, sunan sunadarai: 3-hydroxy-6-methyl-2-ethylpyridine hydrochloride.
Kungiyar magunguna: magungunan hematotropic / antiplatelet, metabolism / antihypoxants da antioxidants, kwayoyinototropic / wakilai na jijiyoyin jini / angioprotector da masu gyaran microcirculation, magunguna na kwayoyin / masu amfani da ophthalmic.
Aikin magunguna: antihypoxic, antiaggregational, antioxidant, angioprotective, retinoprotective.

Kayan magunguna

Methylethylpyridinol sashin angioprotector ne, antihypoxant da antioxidant, yana da kayan aikin retinoprotective. Methylethylpyridinol yana hana matakan tsattsauran ra'ayi kyauta. Methylethylpyridinol yana daidaita sel membranes. Methylethylpyridinol yana inganta microcirculation. Methyl ethyl pyridinol yana rage haɗuwar platelet da dankowar jini, rage jigon ƙwaƙwalwar gaba ɗaya, yana tsawan lokacin coagulation jini, yana haɓaka abubuwan cyclic nucleotides (cyclic guanidine monophosphate da cyclic adenosine monophosphate) a cikin ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwa da platelet. Methylethylpyridinol yana da aikin fibrinolytic, yana ƙarfafa bango na jijiyoyin jiki, rage girman yanayin bango na jijiyoyin jiki da haɗarin basur, yana inganta resorption na basur. Methylethylpyridinol yana daidaita membranes na sel jini da jijiyoyin jini, yana ƙaruwa juriya daga ƙwayoyin jan jini zuwa cutar hemolysis da rauni na injin. Methylethylpyridinol yana ƙaruwa da aiki na enzymes na antioxidant, yana hana isasshen abubuwa masu narkewa na lipids na abubuwan tunawa. Methylethylpyridinol yana da tasirin antitoxic, yana daidaita cytochrome P-450. A cikin matsanancin yanayi, wanda ke haɗuwa da hypoxia da haɓakar liroxidation na lipid, methylethylpyridinol yana haɓaka ayyukan bioenergy. A cikin haɗarin ischemic mai haɗari na ƙwaƙwalwar ƙwayar cuta, methylethylpyridinol yana rage tsananin bayyanar cututtuka, yana ƙaruwa da juriya ga ischemia da hypoxia. Game da haɗarin cerebrovascular (basur da cuta da cuta), methylethylpyridinol yana ba da gudummawa ga gyaran dysfunctions na autonomic, inganta ayyukan mnemonic, da kuma sauƙaƙe maido da ayyukan kwakwalwa. Methylethylpyridinol yana rage samuwar triglycerides, yana da tasirin lipid. Methylethylpyridinol dilates tasoshin jini na zuciya, rage lalacewar ischemic ga myocardium, inganta aikin tsarin motsa zuciya da kwanciyar hankali na zuciya. Methylethylpyridinol yana iyakance girman girman ƙwayoyin necrosis, yana haɓaka matakan sakewa, yana daidaita metabolism na ƙwayar zuciya a cikin infarction myocardial. Methylethylpyridinol yana da tasirin gaske a kan aikin asibiti na infyoction na myocardial, yana rage yiwuwar ciwon zuciya. Game da gazawar jini, methylethylpyridinol yana ba da gudummawa ga tsarin tsarin sake fasalin. Tare da hawan jini, methyl ethyl pyridinol yana da tasirin gaske. Methylethylpyridinol yana kare retina daga lahani na hasken ƙarfi mai ƙarfi, yana inganta microcirculation na ido, kuma yana taimakawa warware matsalar bashin ciki.
Lokacin da aka sanya shi cikin ramin haɗin gwiwa, methylethylpyridinol da sauri ya shiga kyallen fata na ido, inda aka ajiye shi da metabolized. Cigaba da ƙwayar methylethylpyridinol a cikin kyallen ido yana sama da jini. Yana ɗaukar garkuwar jini na jini da kimanin 42%. Tare da gudanarwa na cikin ƙwayar methylethylpyridinol a kashi 10 mg / kg, an lura da ƙarancin rabin rai (minti 18), wanda ke nuna ƙimar kawar da methylethylpyridinol mai yawa daga jini. Maganin cirewar shine minti 0.041. Methylethylpyridinol da sauri ya shiga cikin kyallen takarda da gabobin, inda aka ajiye shi da kuma metabolized. Apparentararren da aka bayyana na rarraba methylethylpyridinol shine lita 5.2. Gabaɗayan aikin methylethylpyridinol shine 214.8 ml / min. An gano metabolites guda biyar, waɗanda ke wakilta ta hanyar samfuran canzawa methylethylpyridinol waɗanda ke rikodin su. Methylethylpyridinol yana cikin metabolized a cikin hanta. An gano mahimmancin 2-ethyl-6-methyl-3-hydroxypyridine-phosphate a cikin hanta. Kwayoyin Methyl ethyl pyridinol metabolites suna dauke da kodan. A cikin yanayin cututtukan cututtukan cuta, alal misali, tare da maganin ƙwaƙwalwa na jijiyoyin jini, canje-canje na magunguna na methylethylpyridinol: haɓakar excretion ta ragu, saboda abin da bioavailability na methylethylpyridinol yana ƙaruwa, lokacin zama na methylethylpyridinol a cikin jini yana ƙaruwa, wanda yana iya zama saboda dawowar sa daga depot, ciki har da ischemic myo.

ischemic bugun jini, bugun jini na jini a cikin lokacin dawowa, rashi na cerebrovascular insufficiency, hadarin mahalli na haihuwar jijiyoyin jiki, sakamakon cerebrovascular da basur da kuma ischemic cerebrovascular accident, rauni na kwakwalwa, rauni na kwakwalwa, postoperative lokaci na epidural da kuma hematomas subdural.
rigakafin cutar rarrabewa, raunin myocardial infarction, angina pectoris ba shi da matsala.
na ciki da ciwan ciki na ciki, zubar jini a farji na cikin ido, basur a cikin ciwan tsofaffi (gami da rigakafin), angioretinopathy (gami da ciwon sankarar mahaifa), dystrophic keratitis, angiosclerotic maculodystrophy (bushe forma, thrombosis, thrombosis, thbobosis) tsakiyar jijiya na retina da rassa, choystretinal dystrophy (gami da maganin chorioretinal dystrophy na asalin atherosclerotic), kariya ta cornea (lokacin sawa x ruwan tabarau) da retina daga fallasa zuwa haske mai tsananin ƙarfi (tare da coagulation na laser, kunar rana da ta ƙonewar laser), cututtukan dystrophic na cornea, rikitarwa na myopia, cataracts (gami da rigakafin kamuwa da mutane a cikin shekaru 40), rauni, kumburi da ƙonewa na cornea, yanayin bayan tiyata dangane da glaucoma tare da maganin choroid, ayyukan tiyata a idanun.

Hanyar yin amfani da methylethylpyridinol da kashi

Ana gudanar da Methylethylpyridinol a cikin cikin ciki, intramuscularly, subconjunctival, parabulbar, retrobulbar, a cikin rami na haɗin gwiwa.
A cikin ramin haɗin gwiwa, kafa 1 zuwa 2 saukad da (bayani 1%) sau 2 zuwa sau 3 a rana, tsawon lokacin kulawa yana dogara da cutar kuma likita yana ƙaddara (yawanci kwanaki 3 zuwa 30), idan an yarda da miyagun ƙwayoyi kuma akwai alamomi, hanya na maganin na iya a ci gaba har zuwa watanni 6 ko maimaita sau 2 zuwa 3 a shekara.
Ana yin Subconjunctival ko parabulbar ana yin sa sau ɗaya a rana ko kuma kowace rana. 0.2 - 0.5 ml na 1% bayani (2 - 5 MG) ana gudanar da subconjunctively, 0.5 - 1 ml na 1% bayani (5 - 10 MG) ana gudanar da shi daidai, tsawon lokacin maganin shine 10 - 30 kwanaki, yana yiwuwa a maimaita a zahiri, idan ya cancanta, sau 2 zuwa 3 a shekara. Idan ya cancanta, ana sarrafa retrobulbar 0.5 zuwa 1 ml na 1% maganin sau ɗaya a rana don kwanaki 10 zuwa 15. Lokacin da coagulation na laser (ciki har da lalata da iyakance coagulation na ciwace-ciwace), retrobulbar ko parabulbar 0.5 zuwa 1 ml na 1% maganin kowace rana da sa'a daya kafin a gudanar da coagulation don kare retina, to 0.5 ml na 1% bayani yana gudana sau ɗaya a rana tsawon kwana 2 zuwa 10.
Angioretinopathy (ciki har da ciwon sukari na angioretinopathy): 0,5 ml parabulbarno (10 mg / ml methylethylpyridinol bayani) sau ɗaya a rana, hanya na maganin shine kwanaki 10. Subconjunctival da jijiyoyin jini na tushen asali daban-daban: parabulbarno ko subconjunctival 0.5 ml (10 mg / ml methylethylpyridinol bayani) sau ɗaya a rana, hanya ta magani shine kwanaki 10-15. Tsarin tsakiya da na yanki na chorioretinal dystrophy, angiosclerotic macular degeneration (bushe bushe): 0,5 ml parabulbarno (methylethylpyridinol bayani 10 mg / ml) sau ɗaya a rana, hanya ta lura shine kwanaki 10-15. Myopia rikice-rikice: 0.5 ml parabulbarno (methylethylpyridinol bayani 10 mg / ml) sau ɗaya a rana, hanya ta magani ita ce kwanaki 10-30, ana iya maimaita hanya sau 2 zuwa 3 a shekara. Thrombosis na tsakiyar jijiya na retina da rassanta: 0,5 ml parabulbarno (methylethylpyridinol bayani 10 MG / ml) sau ɗaya a rana, hanya na maganin shine kwanaki 10-15. Detachment na choroid a cikin marasa lafiya tare da glaucoma a cikin bayan aikin: subconjunctival ko parabulbar 0.5 zuwa 1.0 ml (10 mg / ml methylethylpyridinol bayani) sau ɗaya a kowace kwanaki 2, hanyar kulawa shine injections 10. Cututtukan cututtukan ƙwayar cuta na cornea: subconjunctival 0.5 ml (10 mg / ml methylethylpyridinol bayani) sau ɗaya a rana, hanya na maganin shine kwanaki 10-30. Raunin rauni da ƙonewa na cornea na digiri na biyu: 0,5 ml parabulbarno (methylethylpyridinol bayani 10 mg / ml) sau ɗaya a rana, hanya na maganin shine injections na 10-15.
allura a ciki (20-40 saukad da minti daya), 20-30 ml na maganin 3% (600-900 mg) sau 1 zuwa 3 a rana don kwanaki 5-15, gwargwadon alamun da kuma cutar (pre-diluted da methyl ethyl pyridinol 200 ml na 5% na dextrose ko 0.9% bayani na sodium chloride), to, sun canza zuwa allura ta wucin gadi - 3 zuwa 5 ml na maganin 3% sau 2 zuwa sau 3 a rana tsawon kwanaki 10 zuwa 30.
an gudanar da shi ta hanyar ciki sau 20 (saukad da 20-30 a minti) a cikin kashi 5-10 na MG / kg na kwanaki 10-12, sannan canzawa zuwa allura ta ciki na 2-10 ml (bayani tare da maida hankali na 30 MG / ml) (60-300 mg ) Sau 2 zuwa 3 a rana tsawon kwanaki 10 zuwa 30.
Ana amfani da Methylethylpyridinol a matsayin wani ɓangare na kulawa mai wahala.
Dole ne a gudanar da jiyya tare da methyl ethyl pyridinol a ƙarƙashin kulawar coagulation na jini da tsarin anticoagulation da hauhawar jini.
Idan ya zama dole don amfani da methylethylpyridinol a cikin nau'in ido ya saukad da wasu kwayoyi a cikin hanyar saukad da idanuwa, an sanya methylethylpyridinol daga karshe bayan kammala maganin da ya gabata (aƙalla mintuna 15).
A lokacin jiyya tare da methyl ethyl pyridinol, musamman a gaban nutsuwa, rage karfin jini, ana bada shawara a guji saka hannu cikin ayyukan haɗari waɗanda ke buƙatar haɓakar haɓaka hankali da saurin halayen psychomotor (gami da tuki motocin, hanyoyin).

Haihuwa da lactation

Yin amfani da methylethylpyridinol an hana shi yayin daukar ciki da lactation, tunda babu ingantaccen nazarin ingantaccen binciken lafiyar lafiyar methylethylpyridinol yayin ciki da lactation. Yayin jiyya tare da methyl ethyl pyridinol, ya kamata a dakatar da ciyar da nono.

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