Melfor (Barcelona

Sakamakon yiwuwar haɓaka sakamako mai ban sha'awa, ana ba da shawarar gudanar da maganin capsule. Tafiya da safe. An saita kashi ɗaya akayi daban-daban dangane da alamun da kuma hanyar gudanarwa.
Lokacin ɗauka ta baki, kashi ɗaya shine 0.25-1 g, yawan sarrafawa da tsawon lokacin jiyya yana dogara ne da alamun.
Tare da gudanarwa na iv, kashi ɗaya shine 0.5-1 g 1 lokaci / rana, tsawon lokacin magani yana dogara da alamun.
0.5 ml na allurar bayani tare da maida hankali ne akan 500 MG / 5 ml ana gudanar da shi a cikin layi ɗaya na kwana 10.

Contraindications

Abubuwan kwantar da hankali don amfani da miyagun ƙwayoyi Tafiya sune: karuwar matsin lamba na intracranial (ciki har da lamuran gurbataccen ciki, yawan ciwan ciki), ciki, lactation (shayar da mama), yara da matasa a karkashin shekaru 18, da kara karfin jijiyoyin cutar meldonium.

Yin hulɗa tare da wasu kwayoyi

Lokacin da aka haɗu, meldonium yana haɓaka aikin ƙwayoyin antianginal, wasu magungunan antihypertensive, cardiac glycosides.
Tare da yin amfani da meldonium na lokaci guda tare da nitroglycerin, nifedipine, alpha-blockers, antihypertensive jami'ai da na wurare masu kumburi, tachycardia matsakaici, yanayin jijiya na iya haɓaka (tare da waɗannan haɗuwa, ana buƙatar taka tsantsan).

Alamu don amfani

- Rage yawan aiki, kara yawan motsa jiki, lokacin aikin da ya dace don hanzarta farfadowa.

- A matsayin wani ɓangare na hadaddun farji na cututtukan zuciya da jijiyoyin jiki, gazawar zuciya, ƙwaƙwalwar ƙwayar cuta a kan tushen dishemonal myocardial dystrophy.

- Kamar yadda wani yanki na hadaddun farji don haɗarin cerebrovascular (hadarin cerebrovascular na nau'in ischemic, musamman mahimmin lokaci, ƙarancin ƙwaƙwalwar ƙwayar cuta).

- Cikakken farfaɗo da magani na karbo cutar cututtukan fata.

- Ciwon baya na jijiyoyin jiki, haemophthalmus da bashin jini na kashin baya daban-daban na etiologies, thrombosis daga cikin jijiya na tsakiya da kuma rassan ta, retinopathy na etiologies daban-daban (ciki har da ciwon sukari da hauhawar jini).

Yadda ake amfani: sashi da hanya na jiyya

Magani don allura

Stressara yawan damuwa da ta jiki: a cikin jijiyoyin jini a cikin 500 MG (5 ml) sau ɗaya a rana. Aikin magani shine kwanaki 10-14. Idan ya cancanta, ana maimaita karatun bayan makonni 2-3. Don cututtukan zuciya (a matsayin ɓangare na ƙwaƙwalwar ƙwayar cuta): a cikin kwantar da hankali 500-1000 MG (5-10 ml). Aikin magani shine kwanaki 10-14.

Hadarin Ischemic cerebrovascular, musamman mawuyacin lokaci (a matsayin ɓangare na haɗin haɗuwa): 500 MG cikin ciki (5 ml) 1 lokaci ɗaya kowace rana don kwanaki 7-10, to, ana ɗaukar su a baki.

Rashin ƙwayar ƙwayar cuta na kullum: 500 mg intramuscularly (5 ml) sau ɗaya a rana. Aikin magani shine kwanaki 10-14, sannan sai suka canza zuwa ga baka. Draarfafa ciwo na barasa: cikin jijiyoyin hannu - 500 MG (5 ml) sau 2 a rana. Aikin jiyya shine kwanaki 7-10.

Kwayar cututtukan jijiyoyin jiki na fundus da retinal dystrophy: 50 MG (0.5 ml) maganin allura ana gudanar da aikin retrobulbarly kuma subconjunctively na kwanaki 10.

Ana ɗaukarsa a baki, kafin abinci, saboda sakamako mai ban sha'awa yana da kyau a yi amfani da shi da safe.

Activityara yawan motsa jiki 250 MG sau 4 a rana. Aikin magani shine kwanaki 10-14. Idan ya cancanta, ana maimaita magani bayan makonni 2-3. An tsara 'yan wasan motsa jiki na 500-1000 MG sau 2 a rana kafin horo. Tsawon lokacin karatun a cikin kwanakin shiri shi ne 14-21, a lokacin gasar - kwanaki 10-14.

Tare da cututtuka na zuciya da jijiyoyin jini (a matsayin wani ɓangare na ƙwayar jiyya):

Stress angina pectoris - 250 mg sau 3 a rana don kwanaki 3-4, sannan 250 mg sau 3 a rana sau 2 a mako don watanni 1-1.5.

Myocardial infarction: a cikin lokacin m - cikin jijiyoyi, sannan cikin ciki ta 500 MG kowace rana, ta yin amfani da maganin gaba ɗaya sau ɗaya ko sau 2 a rana.

Rashin ciwon zuciya - 500-1000 MG sau ɗaya a rana. Hanyar magani shine makonni 4-6.

Cardialgia akan tushen dishormonal myocardial dystrophy 250 mg sau 2 a rana. Hanyar magani shine kwana 12.

Hadarin Cerebrovascular: a cikin lokacin m, cikin jijiyoyin jiki, to 500 MG kowace rana, zai fi dacewa a farkon rabin rana. Hanyar magani shine makonni 4-6.

Daukewar cutar barasa (a zaman wani bangare na musamman takamaiman magani) 500 MG sau 4 a rana. Aikin jiyya shine kwanaki 7-10.

Aikin magunguna

Maganin aiki mai aiki da Melfora shine meldonium - analog na roba na gamma-butyrobetaine, wanda ke hana aikin gamma-butyrobetaine hydroxynase. A cikin yanayin ischemia, yana dawo da daidaituwa na tafiyar matakai na isar da oxygen da yawan amfani dashi a sel. Hanyar aiki yana ƙayyade bambancin tasirin magungunansa: haɓaka haɓaka, rage alamun damuwa da damuwa ta jiki, kunna nama da rigakafin ƙwaƙwalwar mutum.

Yana da sakamako mai tasiri: idan akwai mummunan lalacewa na ƙarancin ƙwaƙwalwa na myocardium, rage jinkirin samuwar yankin necrotic, yana gajarta lokacin murmurewa. Tare da rashin karfin zuciya, yana kara yawan kwanciyar hankali na mutum, yana kara karfin motsa jiki, da kuma rage yawan kamuwa da cutar angina. A cikin mummunar cuta da rashin lafiyar ischemic na wurare dabam dabam na haɓakar cerebral yana inganta wurare dabam dabam na jini a cikin ischemia, yana ba da gudummawa ga sake rarraba jini a madadin yankin ischemic. Inganci idan akwai cututtukan jijiyoyin jiki da jijiyoyin ƙwayar cuta dystrophic. Yana da tasirin tonic akan tsarin juyayi na tsakiya kuma yana kawar da rikice-rikice na aiki na tsarin juyayi na somatic da autonomic a cikin marasa lafiya tare da shan barasa tare da ciwo na cirewa.

Side effects

Allergic halayen (redness, fata fatar, itching, kumburi), dyspepsia, tachycardia, rage ko karuwa a cikin jini, tashin hankali ba wuya.

Tare da yawan wuce haddi na Melfort, raguwar hauhawar jini, ciwon kai, tachycardia, dizziness, rauni na gaba ɗaya ke tasowa. Jiyya alama ce.

Nau'i na saki, marufi da abun da ke ciki

KafuraiKafa 1.
meldonium250 MG

5 inji mai kwakwalwa. - fakitin bakin (1) - fakitoci na kwali.
5 inji mai kwakwalwa. - fakitin bakin (2) - fakitoci na kwali.
5 inji mai kwakwalwa. - fakiti mai bakin ciki (3) - fakitoci na kwali.
5 inji mai kwakwalwa. - fakiti mai bakin ciki (4) - fakitoci na kwali.
5 inji mai kwakwalwa. - fakitin bakin (6) - fakitoci na kwali.
5 inji mai kwakwalwa. - fakiti mai bakin ciki (10) - fakitoci na kwali.
10 inji mai kwakwalwa. - fakitin bakin (1) - fakitoci na kwali.
10 inji mai kwakwalwa. - fakitin bakin (2) - fakitoci na kwali.
10 inji mai kwakwalwa. - fakiti mai bakin ciki (3) - fakitoci na kwali.
10 inji mai kwakwalwa. - fakiti mai bakin ciki (4) - fakitoci na kwali.
10 inji mai kwakwalwa. - fakitin bakin (6) - fakitoci na kwali.
10 inji mai kwakwalwa. - fakiti mai bakin ciki (10) - fakitoci na kwali.
30 inji mai kwakwalwa - fakitin bakin (1) - fakitoci na kwali.
30 inji mai kwakwalwa - fakitin bakin (2) - fakitoci na kwali.
30 inji mai kwakwalwa - fakiti mai bakin ciki (3) - fakitoci na kwali.
30 inji mai kwakwalwa - fakiti mai bakin ciki (4) - fakitoci na kwali.
30 inji mai kwakwalwa - fakitin bakin (6) - fakitoci na kwali.
30 inji mai kwakwalwa - fakiti mai bakin ciki (10) - fakitoci na kwali.
10 inji mai kwakwalwa. - polymer kwantena (1) - fakitoci na kwali.
Guda 20. - polymer kwantena (1) - fakitoci na kwali.
30 inji mai kwakwalwa - polymer kwantena (1) - fakitoci na kwali.
Guda 40. - polymer kwantena (1) - fakitoci na kwali.
Guda 50. - polymer kwantena (1) - fakitoci na kwali.
Guda 100 - polymer kwantena (1) - fakitoci na kwali.

Alamar magunguna

Don maganin baka ko na cikin jijiya: a matsayin wani ɓangare na hadaddun farjin cututtukan zuciya na zuciya (angina pectoris, myocardial infarction), raunin zuciya, rashin tausayi na zuciya, dishormonal cardiomyopathy, a matsayin wani ɓangare na hadaddiyar farfaɗar cututtukan cututtukan ƙwaƙwalwa da rashin rikicewar ƙwayar cuta (bugun jini da rashin ƙwaƙwalwar ƙwayar cuta), rage aiki, ƙarancin jiki (ciki har da a cikin 'yan wasa), bayan aikin da ya dace don hanzarta farfadowa, cire ciwo a cikin shan barasa (a hade tare da takamaiman aikin likita, barasa ZMA).

Don gudanar da tsarin parabulbar: rikicewar yanayin jijiyoyin jini a cikin retina, hemophthalmus da cututtukan fata na kashin baya daban-daban na etiologies, thrombosis na jijiya na tsakiya da reshenta, retinopathy na etiologies daban-daban (ciki har da masu ciwon sukari da hauhawar jini) - kawai don maganin parabulbar.

Lambobin ICD-10
Lambar ICD-10Nuna
F10.3Karbo jihar
H34Kasancewa na Jijiyoyin bugun ciki
H35.0Fassarar fata da kuma canje-canje na jijiyoyin jiki
H35.6Kwakwalwar koda
H36.0Rashin maganin ciwon sukari
H44.8Sauran cututtuka na ƙwallon ido (ciki har da haemophhalmus)
I20Angina pectoris
I21Babban myocardial infarction
I42Cardiomyopathy
I50.0Ciwon Zuciya
I61Cutar ciki na ciki (nau'in basur na nakasar ciki)
I63Cerbral infarction
Z54Jihar dawo da
Z73.0Aikuwa
Z73.3Halin damuwa ba a rarraba shi wani wuri (damuwa na jiki da kwakwalwa)

Sakawa lokacin

Dangane da yiwuwar haɓaka sakamako mai ban sha'awa, ana bada shawara don amfani dashi da safe. An saita kashi ɗaya akayi daban-daban dangane da alamun da kuma hanyar gudanarwa.

Lokacin ɗauka ta baki, kashi ɗaya shine 0.25-1 g, yawan sarrafawa da tsawon lokacin jiyya yana dogara ne da alamun.

Tare da gudanarwa na iv, kashi ɗaya shine 0.5-1 g 1 lokaci / rana, tsawon lokacin magani yana dogara da alamun.

0.5 ml na allurar bayani tare da maida hankali ne akan 500 MG / 5 ml ana gudanar da shi a cikin layi ɗaya na kwana 10.

Umarni na musamman

Yi amfani tare da taka tsantsan a cikin cututtukan hanta da / ko kodan, musamman na dogon lokaci.

Shekaru da yawa na gogewa a cikin lura da matsanancin ƙwayar cuta na zuciya da rashin angina a cikin sassan aikin zuciya yana nuna cewa meldonium ba shine farkon layin farko na cututtukan jijiyoyin zuciya ba.

Hulɗa da ƙwayoyi

Lokacin da aka haɗu, meldonium yana haɓaka aikin ƙwayoyin antianginal, wasu magungunan antihypertensive, cardiac glycosides.

Tare da yin amfani da meldonium na lokaci guda tare da nitroglycerin, nifedipine, alpha-blockers, antihypertensive jami'ai da na wurare masu kumburi, tachycardia matsakaici, yanayin jijiya na iya haɓaka (tare da waɗannan haɗuwa, ana buƙatar taka tsantsan).

Hanyar aikin

Magungunan kwatancin ɗan adam ne na γ-butyrobetaine. Yana da tasiri mai yawa a cikin hadaddun carnitine da motsi mai acid ta hanyar bangon tantanin halitta, kuma yana hana tarin abubuwan da ake samu na acetyl coenzyme da acyl carnitine a cikin sel.

Pharmacodynamics na miyagun ƙwayoyi ya ƙunshi haɓaka matakin aikin.

A cikin lura da ischemia, miyagun ƙwayoyi suna daidaita yanayin jigilar / amfani da oxygen ta sel, yana hana motsi na ATP kuma yana kunna glycolysis. Ta hanyar rage matakin carnitine, ƙwayar tana inganta wurare dabam dabam na gamma-butyrobetaine, wanda ke da tasirin vasodilating. Magungunan ƙwayar magunguna sun haɗa da haɓaka matakin aiki, rage girman tasirin damuwa na jiki / hankali, da inganta rigakafin ƙwayoyin cuta / ƙwayar nama.

A cikin manyan siffofin ischemia, miyagun ƙwayoyi yana hana ƙarancin kwanciyar hankali da ayyukan necrotic, tare da hanzarta farfadowa. Bugu da kari, sautunan tsakiya na jijiyoyin jiki kuma suna aiwatar da aiki a alamu na cire barasa.

Ana samun maganin daga hanjin. Its bioavailability ya kai 78%.

Matsakaicin maida hankali bayan kulawa ta baka an lura dashi bayan minti 60-120.

A lokacin biotransformation, da miyagun ƙwayoyi samar da wani biyu daga metabolites a cikin jiki. Cire rabin rayuwar shine daga 3 zuwa 6 hours. Kodan ya fitar da maganin.

Abun ciki da nau'i na saki

A kan siyarwa, ana ba da maganin ta hanyar capsules da maganin allura.

Kwaya 1 ta ƙunshi:

  • kashi na aiki (meldonium dihydrate) - 500 MG,
  • sauran aka gyara: 27.2 MG na dankalin turawa, sittin, 10.8 mg na sillofon silicon dioxide, 5.4 MG na alli stearate,
  • jikin kwalliya da kwalliya sune gelatin 98% da 2% titanium dioxide.

A cikin capsules farin farin hygroscopic foda ne.

A kan siyarwa, ana ba da magani a cikin nau'i na capsules.

An sanya mafita a cikin ampoules 5 ml, waɗanda suke cikin fakiti na katako da akwatunan kwali.

Side effects

Ayyukan jiki na gaba ga miyagun ƙwayoyi suna yiwuwa:

  • rashin lafiyan: kumburi, kurji, jan launi (mafi wuya),
  • Gastrointestinal fili: bayyanuwar cutar dyspeptik,
  • CNS: ƙarfafawar halayen psychomotor,
  • CVS: karuwa / raguwa a cikin karfin jini, tachycardia (a cikin matsanancin yanayi).

Bayan amfani da miyagun ƙwayoyi, kurji yana yiwuwa.

Amfani da barasa

Abubuwan da ke amfani da maganin sun bayyana a cikin kusan awa 12. Bayan wannan lokacin, haɗarin mummunan halayen hulɗa da miyagun ƙwayoyi tare da sauran abubuwan ba ya nan ko ƙananan ƙananan.

Umarni game da amfani da miyagun ƙwayoyi bai hana a hada shi da giya ba. Koyaya, idan tafarkin gudanarwarsa zai gudana don kula da kowace cuta ta tsarin zuciya ko haɗarin cerebrovascular, mai haƙuri ya kamata ya guji amfani da barasa. Wannan ya faru ne sakamakon haɗarin raguwa a cikin ayyukan magungunan ƙwayoyi. Haɗin kai ɗaya na iya haifar da:

  • mummunan bayyanar rashin lafiyar,
  • tachycardia da angina pectoris,
  • yanayin dyspeptik
  • tsalle a cikin karfin jini.

Lokacin shan magani da barasa, tsalle-tsalle cikin karfin jini na iya bayyana.

Ranar karewa

Ba a wuce shekaru 4 ba daga ranar samarwa. Haramun ne a sha kuma a sa magani, ranar karewa wanda ya ƙare.

Wani lokaci, idan magani ba ya nan ko bai dace ba saboda contraindications, zaku iya kula da maye gurbin sa.

Mafi inganci kuma sanannun su sune:

Sakamakon rashin halayen marasa kyau yayin gudanarwa da tasiri, ƙwayar tana karɓar yawancin maganganu masu inganci daga likitoci da masu haƙuri. Yana ba da gudummawa don haɓaka haɓakawa da kuma dawo da makamashi.

Gennady Oprishchenko (therapist), dan shekara 40, Pushkino

Dukkan nau'ikan magungunan (capsules da bayani) suna daidai da tasiri a cikin alamun cirewa, rikicewar jijiyoyin jini a cikin GM da sauran cututtukan cuta. Marasa lafiya sun gamsu da araha a farashin magani da kusan kusan babu "sakamako masu illa".

Ekaterina Kolpakova (therapist), dan shekara 36, ​​Yaroslavl

Ina rubuto magani ne ba kawai ga marassa lafiya ba, har ma da lafiyar mutane (masu motsa jiki) don inganta aikin. Zai taimaka sosai idan aka doru a kan matsanancin damuwa da damuwa a jiki. Abubuwan da ke haifar da sakamako masu illa na tsawon lokacin aikina ba su taɓa gani ba.

Stanislav Smirnov, mai shekara 41, Ryazan

Magungunan sun taimaka wa ɗan'uwana ya warke daga shan giya. Likita ya umarta a hade tare da sauran allunan. Yanzu ɗan'uwan ya sami aiki kuma yana jagorantar rayuwa mai kyau.

Inga Stepanenko, 38 years old, Sergiev Posad

Magungunan ya bugu ne yayin da ya kasa samun nasara a cikin gudanawar kwakwalwa. Ynamarfafa aiki yana bayyana da sauri, raunin sakamako masu illa yana iya faruwa sai dai yin farin ciki. Ee, kuma farashin mai araha ne.

Melfor haƙuri sake dubawa

Likita ya umurce ni da Melfor a matsayin ƙyalli analog na wani magani. Don haka ya tambaye ni - don rubuta magani mai tsada ko maras tsada na gida.Me yasa nake buƙatar shigo da tsada? Watanni da yawa yanzu, an wajabta mani kuma akwai wani tasiri: ya zama da sauƙin yin tafiya, angina harin ba shi da haɗari. Gaba ɗaya, na yi farin ciki da Melfor sosai. Godiya ta musamman ga likitocin da suka fahimci cewa wadanda suka yi ritaya na iya samun kudi don magunguna masu tsada da aka shigo da su kuma ba su zabi su yi!

Short Short

Maganin kwantar da tarzoma a cikin gida shine magani na Melfor (ƙwayar meldonium mai aiki) - magani ne na rayuwa wanda ke motsa ƙoshin tafiyar matakai da inganta haɓaka samar da kyallen takarda. Yana hana shigarwar zuwa cikin mitochondria na kitse mai kyauta, ta haka ne zai rage adadin kuzari na karshen. Melfore yana ƙuntata zirga-zirgar mai mai ta hanyar membranes na mitochondrial, duk da haka, yana aiki a wannan batun mai zaɓar, ba kawai yana ƙaddamar da mayuka mai ɗorewa ba. Amma ga gajeren sarkar, zasu iya shiga cikin mitochondria kuma suyi duk abin da suke so a can (da farko, muna magana ne game da iskar shaye shaye). Ba kamar na trimetazidine ba, Melfore ba ya haifar da tara ƙwayoyin kitse mai ƙarfi a cikin mitochondria. A ƙarshen asalin ischemia, ƙwayar ta dawo da daidaitacciyar daidaituwa a cikin ayyukan jigilar oxygen zuwa kyallen da kuma yawan amfani da shi a wuraren bayarwa. A lokaci guda, anaerobic glycolysis yana ƙaruwa. A karkashin aikin melphor, gamma-butyrobetaine vasodilator ya fara rayayye. Magungunan yana inganta aikin, a hankali yana rage alamun gajiya ta jiki da ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwa, yana inganta yanayin rigakafi, yana aiki akan duka ƙwayoyin salula da ƙwaƙwalwar mutum, kuma yana da sakamako na zuciya. A cikin mummunan ischemic lalacewar ƙwayar zuciya, Melfor yana rage girman ƙwanƙolin ƙwaƙwalwar ƙwayar ƙwaƙwalwa, yana hanzarta farfadowa. Tare da rashin isasshen aikin zuciya, yana kara kwarjinin kwarin gwiwar zuciya, da inganta haqurin motsa jiki, da rage hadarin angina pectoris. Tare da ischemia na cerebral, melfor yana inganta hawan jini a cikin ischemic foci, yana jagorantar kwararar jini da farko zuwa yankunan ischemic. Ba wanda zai iya kasa fahimtar fa'idar fa'idar amfani da Melfor don cututtuka na asusus (jijiyoyin bugun gini da dystrophic).

Hakanan za'a iya amfani da miyagun ƙwayoyi a cikin hadaddun kulawa da marasa lafiya da ke fama da rashin shan giya mai kwakwalwa: yana yin amfani da tsarin juyayi na tsakiya kuma yana kawar da tasirin rikicewar aiki a ɓangaren sa. Jerin tasirin sakamako mai kyau na Melfor bai iyakance ga wannan ba: alal misali, maganin yana nuna sakamako na antioxidant, hana peroxidation na lipid da kunna antioxidant na antioxidants, sakamakon abin da sakamakon damuwa na oxidative ya ragu. A cikin karatun asibiti, an tabbatar da ikon Melfor don yin tasiri ga ayyukan endothelium da daidaita sautin jijiyoyin jini. Bugu da kari, an gano cewa miyagun ƙwayoyi shima yana da sauran tasirin jijiyoyin jini: alal misali, yana kawar da jijiyoyin bugun jini adresal da angiotensin, kuma yana rage juriya na gaba ɗaya na jijiyoyin bugun jini. Bugu da kari, melfor yana kara karfin jijiyoyin jikin mutum zuwa insulin, yana sarrafa metabolism na lipids da glucose.

Melfor yana samuwa a cikin siffofin sashi biyu: capsules da bayani don allura. Yana da kyau a sha maganin da safe, kamar yadda zai iya zama mai ban sha'awa. Ana saita maganin ta likita daban daban. Dangane da shawarar gabaɗaya don gudanar da maganin magana, kashi ɗaya na Melfor shine 0.25-1 g, yawan sarrafawa da tsawon lokacin karatun miyagun ƙwayoyi an ƙaddara shi ta takamaiman alamun. Tare da gudanarwa na ciki, kashi na yau da kullum na miyagun ƙwayoyi shine 0.5-1 g, ana gudanarwa a lokaci guda. Parabulbar (ta hanyar fata na ƙananan fatar ido) Ana gudanar da Melfor a cikin 0.5 ml na kwanaki 10. A ƙarshe, muhimmiyar sanarwa: kamar yadda karatun asibiti da ƙwarewa a jiyya na angina mai rashin ƙarfi da rashin ƙarfi mai zurfi ya nuna, Melfor ba shine farkon zaɓi a cikin ciwo na rashin jijiya ba.

Pharmacology

Hanyoyin haɓaka ƙwayar cuta, anama gamma-butyrobetaine. Yana hana gamma-butyrobetaine hydroxynase, yana hana haɗarin carnitine da jigilar daskararren sarkar acid ta hanyar membranes, kuma yana hana tara nau'ikan kitse mai ɗorewa a cikin sel - abubuwan da ake kira acylcarnitine da acylcoenzyme A.

A karkashin yanayin ischemia, yana dawo da daidaituwa na tafiyar matakai na isar da oxygen da yawan amfani da shi a cikin sel, yana hana cin zarafin jigilar jirgin ATP, kuma a lokaci guda yana kunna glycolysis, wanda ke gudana ba tare da ƙarin amfani da oxygen ba. Sakamakon raguwa a cikin taro na carnitine, gamma-butyrobetaine tare da kaddarorin vasodilating yana haɓaka mai ƙarfi. Hanyar aiki yana ƙayyade bambancin tasirin magunguna: haɓaka haɓaka, rage alamun damuwa da damuwa na jiki, kunna nama da rigakafin ƙwaƙwalwar mutum, tasirin cutar zuciya.

Game da mummunar cutar ischemic a cikin myocardium, yana rage jinkirin samuwar yankin necrotic kuma yana gajarta lokacin murmurewa. Tare da rashin karfin zuciya, yana kara yawan kwanciyar hankali na mutum, yana kara karfin motsa jiki, da kuma rage yawan kamuwa da cutar angina. A cikin mummunar cuta da rashin lafiyar ischemic na wurare dabam dabam na haɓakar cerebral yana inganta wurare dabam dabam na jini a cikin ischemia, yana ba da gudummawa ga sake rarraba jini a madadin yankin ischemic. Inganci ga cututtukan jijiyoyin bugun gini da na dystrophic na fundus. Yana da sakamako na tonic akan tsarin juyayi na tsakiya, yana kawar da rikice-rikice na aiki na tsarin juyayi a cikin marasa lafiya tare da shan barasa tare da ciwo na cirewa.

Pharmacokinetics

Bayan gudanar da baki, yana sha da sauri daga narkewa. Bioavailability kusan kashi 78%. Cmax a cikin plasma ana samun sa'o'i 1-2 bayan gudanarwa. An yi shi a cikin jiki tare da samuwar manyan abubuwan metabolites guda biyu waɗanda kodan ke bankwana da su. T1/2 shine 3-6 hours kuma ya dogara da kashi.

Haɗin kai na Melfor tare da wasu kwayoyi

Hatsarin haɓakar jijiyoyin jini da tachycardia matsakaici na faruwa ne sakamakon amfanin Melfort na lokaci guda tare da kwayoyi masu zuwa:

  • na kewaye vasodilators,
  • alfa talla
  • antihypertensive jami'ai
  • nifedipine
  • nitroglycerin.

Bugu da ƙari, idan aka haɗo su tare da glycosides cardiac, magungunan antianginal, da kuma wasu nau'ikan magungunan antihypertensive, tasirin su yana daɗaɗawa.

Yawan abin sama da ya kamata

Game da shan magunguna masu yawa, jin rauni na gaba daya, ciwon kai da farin ciki, haɓakar tachycardia, da raguwar hauhawar jini. Tunda wannan magani yana da guba mai guba, duk bayyananniyar bayyanannun takan lalace cikin sauri bayan daidaitaccen maganin cutar siga.

Sharuɗɗan da yanayin ajiya

Rayuwar shiryayye na miyagun ƙwayoyi Melfor shine watanni 24 daga ranar da aka sake su. Kiyaye shi a cikin busassun wuri mai duhu mara amfani ga yara.

Yanayin zafin jiki kada ya wuce +25 digiri Celsius.

Ana samun magungunan Melfor a cikin magunguna. Matsakaicin matsakaicinta a Rasha shine 500-560 rubles.

A cikin magunguna na Yukren Kuna iya siyan magani na Melfor akan farashi hryvnia 200 zuwa 250.

A wasu halaye, idan miyagun ƙwayoyi Melfor bai dace ba, ko kuma ba za a samu damar amfani da shi ba, ya kamata ku kula da mafi kyawun musanyawa.

Shahararrun analogues na Melfora sun hada da:

  • Magnikor - wani shiri ne da ya danganta da Acetylsalicylic acid da magnesium hydroxide, wadanda aka yi niyya don magance cututtukan zuciya da na jijiyoyin jiki da kuma kamuwa da cuta,
  • Pumpan - magani a cikin hanyar saukad da Allunan don hadadden lura da jijiya hauhawar jini, zuciya rashin cin nasara, arrhythmia da wasu sauran cututtukan zuciya,
  • Cordaflex - Allunan za'a iya cinye shi suna dauke da babban sinadarin nifedipine. An tsara wannan magani don tsayayyen angina pectoris, tashin hankali na hauhawar jini, cututtukan zuciya da jijiyoyin jini, da hauhawar jijiyoyin jini, wanda ke da tsananin wahala,
  • Corvitol - allunan dauke da metoprolol. Ana amfani dasu don maganin cututtukan zuciya da jijiyoyin jini, infarction na zuciya na zuciya, jijiyoyin jini, cututtukan zuciya, hawan jini, da kuma cututtukan zuciya,
  • Kudesan magani ne a cikin nau'ikan saukad da alluna dangane da ubidecarinone. Babban alamomi game da amfaninsu shine cututtukan zuciya da na zuciya, gazawar zuciya, arrhythmia, da kuma lokacin dawowa bayan fama da rauni na zuciya,
  • Amlipin magani ne mai hade dangane da lisinopril da amlodipine, wanda aka yi niyya don magance cututtukan zuciya da jijiyoyin jini da kuma tsananin raunin jiki,
  • Bisoprol - allunan da ke kan furucin bisoprol, an yi niyya don maganin angina pectoris, gajiyawar zuciya, da kuma hauhawar jini.

Sakamakon babban tasiri da rashin halayen sakamako, miyagun ƙwayoyi Melfor suna karɓar ingantaccen dubawa daga marasa lafiya da likitoci. Ana samun cikakkun bayanai a ƙarshen wannan labarin.

Mutanen da suka sha maganin sun lura yana da fa'ida ga tsarin jijiyoyin zuciya da kuma aikin jijiyoyin jini. Hakanan yana ba da gudummawa ga saurin dawo da ƙarfi da haɓaka haɓaka.

Idan kuna da kwarewar kanku game da magani tare da amfani da miyagun ƙwayoyi Melfor, tabbatar da cewa ku raba ra'ayinku tare da sauran baƙi zuwa shafin, barin sake bita.

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